Privileged scaffolds for library design and drug discovery

The evolving role of natural products in drug discovery

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Target-Oriented and Diversity-Oriented Organic Synthesis in Drug Discovery

Schreiber, S. L. (2000) · Science · doi:10.1126/science.287.5460.1964 · Cited by 2,571

Drugs for bad bugs: confronting the challenges of antibacterial discovery

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A Planning Strategy for Diversity‐Oriented Synthesis

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Methods for drug discovery: development of potent, selective, orally effective cholecystokinin antagonists

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Exploiting Chemical Libraries, Structure, and Genomics in the Search for Kinase Inhibitors

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From Nature to Drug Discovery: The Indole Scaffold as a ‘Privileged Structure’

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Diversity-oriented synthesis: Exploring the intersections between chemistry and biology

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Privileged Structures: Applications in Drug Discovery

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Towards the Optimal Screening Collection: A Synthesis Strategy

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Synthesis of Tetrahydroquinoline‐Embedded Bridged Benzothiaoxazepine‐1,1‐dioxides

Borgohain, H., Devi, R., Dheer, D., Borah, B. J., Shankar, R., & Das, S. K. (2017) · European Journal of Organic Chemistry · doi:10.1002/ejoc.201701152 · Cited by 21

Regioselective Reaction of HeterocyclicN-Oxides, an Acyl Chloride, and Cyclic Thioethers

Frei, P., Jones, D. H., Kay, S. T., McLellan, J. A., Johnston, B. F., Kennedy, A. R., & Tomkinson, N. C. O. (2018) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.7b02457 · Cited by 21

Rhodium(III)-Catalyzed Synthesis of Spiropiperidine Derivatives via C–H Activation

Péneau, A., Retailleau, P., Guillou, C., & Chabaud, L. (2018) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.7b03252 · Cited by 21

Effect of N-1 arylation of monastrol on kinesin Eg5 inhibition in glioma cell lines

Gonçalves, I. L., Rockenbach, L., das Neves, G. M., Göethel, G., Nascimento, F., Kagami, L. P., Figueiró, F., de Azambuja, G. O., Dias, A. D. F., Amaro, A., et al. (2018) · MedChemComm · doi:10.1039/c8md00095f · Cited by 21

Mesoporous silica supported ytterbium as catalyst for synthesis of 1,2‐disubstituted benzimidazoles and 2‐substituted benzimidazoles

Samanta, P. K., Banerjee, R., Richards, R. M., & Biswas, P. (2018) · Applied Organometallic Chemistry · doi:10.1002/aoc.4507 · Cited by 21

Benzimidazole

Singh, P. K., & Silakari, O. (2018) · Elsevier eBooks · doi:10.1016/b978-0-08-102083-8.00002-9 · Cited by 21

Facile synthesis of thiochromeno[2,3-b]indol-11(6H)-ones and pyrido[3′,2′:5,6]thiopyrano[2,3-b]indol-5(10H)-ones

Kiamehr, M., Moghaddam, F. M., Semeniuchenko, V., Villinger, A., Langer, P., & Iaroshenko, V. O. (2013) · Tetrahedron Letters · doi:10.1016/j.tetlet.2013.07.012 · Cited by 21

Effect of isoxazole derivatives of tetrahydrofuran neolignans on intracellular amastigotes of Leishmania (Leishmania) amazonensis: A structure–activity relationship comparative study with triazole‐neolignan‐based compounds

das Neves, A. R., Trefzger, O. S., Barbosa, N. V., Honorato, A. M., Carvalho, D. B., Moslaves, I. S. B., Toffoli-Kadri, M. C., Yoshida, N., Kato, M. J., de Arruda, C. C. P., et al. (2019) · Chemical Biology & Drug Design · doi:10.1111/cbdd.13609 · Cited by 21

Rhodium-Catalyzed Diastereo- and Enantioselective Tandem Spirocyclization/Reduction of 3-Allenylindoles: Access to Functionalized Vinylic Spiroindolines

Grugel, C. P., & Breit, B. (2019) · Organic Letters · doi:10.1021/acs.orglett.9b03835 · Cited by 21

Enantioselective Synthesis of α‐Secondary and α‐Tertiary Piperazin‐2‐ones and Piperazines by Catalytic Asymmetric Allylic Alkylation

Korch, K. M., Eidamshaus, C., Behenna, D. C., Nam, S., Horne, D. A., & Stoltz, B. M. (2014) · Angewandte Chemie · doi:10.1002/ange.201408609 · Cited by 21

Identification of strategic molecules for future circular supply chains using large reaction networks

Weber, J. M., Lió, P., & Lapkin, A. A. (2019) · Reaction Chemistry & Engineering · doi:10.1039/c9re00213h · Cited by 22

Lead selection of antiparasitic compounds from a focused library of benzenesulfonyl derivatives of heterocycles

Pagliero, R. J., Kaiser, M., Brun, R., Nieto, M. J., & Mazzieri, M. R. (2017) · Bioorganic & Medicinal Chemistry Letters · doi:10.1016/j.bmcl.2017.07.081 · Cited by 21

Substituted tetrahydroisoquinolines: synthesis, characterization, antitumor activity and other biological properties

Capilla, A. S., Soucek, R., Grau, L., Romero, M., Rubio, J., Caignard, D. H., & Pujol, M. D. (2018) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2017.12.098 · Cited by 21

Neuroprotective Potential of Indole-Based Compounds: A Biochemical Study on Antioxidant Properties and Amyloid Disaggregation in Neuroblastoma Cells

Ciaglia, T., Miranda, M. R., Micco, S. D., Vietri, M., Smaldone, G., Musella, S., Sarno, V. D., Auriemma, G., Sardo, C., Moltedo, O., et al. (2024) · Antioxidants · doi:10.3390/antiox13121585 · Cited by 20

Hydroamination of alkenyl N-arylhydrazones mediated by t-BuOK for the synthesis of nitrogen heterocycles

Peng, X., Kaga, A., Hirao, H., & Chiba, S. (2016) · Organic Chemistry Frontiers · doi:10.1039/c6qo00053c · Cited by 20

Exploration of synthetic multifunctional amides as new therapeutic agents for Alzheimer's disease through enzyme inhibition, chemoinformatic properties, molecular docking and dynamic simulation insights

Hassan, M., Abbasi, M. A., Rehman, A.-U., Siddiqui, S. Z., Hussain, G., Shah, S. A. A., Shahid, M. A. R., & Seo, S. (2018) · Journal of Theoretical Biology · doi:10.1016/j.jtbi.2018.09.018 · Cited by 20

Metal-, Photocatalyst-, and Light-Free Minisci C–H Acetylation of N-Heteroarenes with Vinyl Ethers

Dong, J., Liu, J., Song, H., Liu, Y., & Wang, Q. (2021) · Organic Letters · doi:10.1021/acs.orglett.1c01310 · Cited by 20

HFIP-mediated three-component imidization of electron-rich arenes with in situ formed spiroindolenines for facile construction of 2-arylspiroindolenines

Ge, C., Wang, L., Hu, F., Ding, Z., Li, X., Xiao, D., Wang, J., & Li, S. (2022) · Organic Chemistry Frontiers · doi:10.1039/d1qo01862k · Cited by 20

Desulfinative Alkylation of Heteroarenes via an Electrostatic Electron Donor–Acceptor Complex

Laha, R., Patel, T. I., & Moschitto, M. J. (2022) · Organic Letters · doi:10.1021/acs.orglett.2c02932 · Cited by 20

Metal complexes of xanthine and its derivatives: Synthesis and biological activity

Dar, M. O., Mir, R. H., Mohi-ud-din, R., Masoodi, M. H., & Sofi, F. A. (2023) · Journal of Inorganic Biochemistry · doi:10.1016/j.jinorgbio.2023.112290 · Cited by 20

Green synthesis of new quinolinoquinazoline derivatives via one‐pot multicomponent reactions using ZnO / TiO2 @ MWCNTs as a new nanocatalyst

Hasani, L., Ezzatzadeh, E., & Hossaini, Z. (2023) · Journal of Heterocyclic Chemistry · doi:10.1002/jhet.4733 · Cited by 20

Design and synthesis of chromene-1,2,3-triazole benzene sulfonamide hybrids as potent carbonic anhydrase-IX inhibitors against prostate cancer

Albelwi, F. F., Nafie, M. S., Albujuq, N. R., Hourani, W., Aljuhani, A., Darwish, K. M., Tawfik, M. M., Rezki, N., & Aouad, M. R. (2024) · RSC Medicinal Chemistry · doi:10.1039/d4md00302k · Cited by 20

Primary amino acid catalyzed asymmetric intramolecular Mannich reaction for the synthesis of 2-aryl-2,3-dihydro-4-quinolones

Mondal, B., & Pan, S. C. (2014) · Organic & Biomolecular Chemistry · doi:10.1039/c4ob02146k · Cited by 20

Synthesis of novel molecular probes inspired by harringtonolide

Hegde, V. S., Campitelli, M. R., Quinn, R. J., & Camp, D. (2011) · Organic & Biomolecular Chemistry · doi:10.1039/c1ob05299c · Cited by 20

A General Way to Construct Arene‐Fused Seven‐Membered Nitrogen Heterocycles

Bakulina, O., Chizhova, M., Dar’in, D. V., & Krasavin, M. (2017) · European Journal of Organic Chemistry · doi:10.1002/ejoc.201701642 · Cited by 20

Temperature-Controlled Thiation of α-Cyano-β-Alkynyl Carbonyl Derivatives for De Novo Synthesis of 2-Aminothiophenes and Thieno[2,3-c]isothiazoles

Kao, T., Peng, P.-K., Liang, M.-C., Lee, C., Chen, I., Shia, K., & Wu, Y. (2018) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.8b01866 · Cited by 20

Minisci‐Type C–H Cyanoalkylation of Heteroarenes Through N–O/C–C Bonds Cleavage

Jian, Y., Chen, M., Yang, C., & Xia, W. (2019) · European Journal of Organic Chemistry · doi:10.1002/ejoc.201900406 · Cited by 20

Synthesis and anticancer activity of N-9- and N-7- substituted 1,2,3 triazole analogues of 2,6-di-substituted purine

Khazir, J., Mir, B. A., Chashoo, G., Pilcher, L. A., & Riley, D. L. (2019) · Medicinal Chemistry Research · doi:10.1007/s00044-019-02456-9 · Cited by 20

Metal‐free Photocatalytic Intermolecular anti‐Markovnikov Hydroamination of Unactivated Alkenes

Zhao, G., Li, J., & Wang, T. (2021) · European Journal of Organic Chemistry · doi:10.1002/ejoc.202100049 · Cited by 20

A multicomponent tetrazolo indole synthesis

Lei, X., Lampiri, P., Patil, P., Angeli, G. K., Neochoritis, C. G., & Dömling, A. S. S. (2021) · Chemical Communications · doi:10.1039/d1cc02384e · Cited by 20

Copper-catalyzed amino radical tandem cyclization toward the synthesis of indolo-[2,1- a ]isoquinolines

Liu, M., Wang, J., Li, X.-S., Sun, W., & Liu, X. (2022) · Organic Chemistry Frontiers · doi:10.1039/d2qo00051b · Cited by 20

Single step incorporation of isatin to enaminone: a recyclable catalyst towards assembly of diverse four ring fused pyrrolo[2,3,4-kl]acridin-1-ones

Li, C., & Zhang, F. (2016) · RSC Advances · doi:10.1039/c6ra18048e · Cited by 20

Synthesis and evaluation of the anti-proliferative activity of diaryl-3-pyrrolin-2-ones and fused analogs

Mowery, P., Mejia, F. B., Franceschi, C. L., Kean, M. H., Kwansare, D. O., Lafferty, M. M., Neerukonda, N. D., Rolph, C. E., Truax, N. J., & Pelkey, E. T. (2016) · Bioorganic & Medicinal Chemistry Letters · doi:10.1016/j.bmcl.2016.11.076 · Cited by 20

Formulation of benzoxaborole drugs in PLLA: from materials preparation to in vitro release kinetics and cellular assays

Sene, S., McLane, J. S., Schaub, N. J., Bégu, S., Mutin, P. H., Ligon, L. A., Gilbert, R. J., & Laurencin, D. (2015) · Journal of Materials Chemistry B · doi:10.1039/c5tb02258d · Cited by 19

Green and efficient synthesis of 2, 3-dihydroquinazolin-4(1H)-ones in aqueous medium using ZnFe2O4 catalyst under microwave irradiation

Rupnar, B. D., Kachave, T. R., Patil, P. D. J., Shisodia, S. U., & Pawar, R. P. (2017) · Journal of the Iranian Chemical Society · doi:10.1007/s13738-017-1124-y · Cited by 19

Substituent Enabled Divergent Synthesis of N‐Heterocycles: a Metal Carbene Approach Involving Intramolecular Carbene Interception

Xu, H., Xü, K., Jia, Z., Zhou, H., Jiang, P., Lu, X., Pan, Y., Wu, H., Ding, Y., Shen, M., et al. (2014) · Asian Journal of Organic Chemistry · doi:10.1002/ajoc.201402151 · Cited by 19

Three-in-one: information encryption, anti-counterfeiting and LD-tracking of multifunctional purine derivatives

Wang, H., Yu, K., Tan, C.-Y., Li, K., Liu, Y., Shi, L., Lü, K., & Yu, X. (2021) · Journal of Materials Chemistry C · doi:10.1039/d0tc05221c · Cited by 18

Synthesis, Molecular Docking Analysis and in Vitro Biological Evaluation of Some New Heterocyclic Scaffolds-Based Indole Moiety as Possible Antimicrobial Agents

Hassan, E. A., Shehadi, I. A., Elmaghraby, A. M., Mostafa, H. M., Zayed, S. E., & Abdelmonsef, A. H. (2022) · Frontiers in Molecular Biosciences · doi:10.3389/fmolb.2021.775013 · Cited by 19

Synthesis of Pyrazolo[1,5-a]pyridinyl, Pyrazolo[1,5-a]quinolinyl, and Pyrazolo[5,1-a]isoquinolinyl Sulfonyl Fluorides via a [3 + 2] Annulation

Wu, W., & Qin, H. (2023) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.2c02242 · Cited by 19

Intramolecular Arene C(sp 2 )–H Amidation Enabled by Ferrocenium-Mediated Decomposition of 1,4,2-Dioxazol-5-ones as Amidyl Radical Precursors

Sun, W., Au, C., Wong, K.-W., Chan, K. L., Ngai, C. K., Lee, H. K., Lin, Z., & Yu, W. (2023) · ACS Catalysis · doi:10.1021/acscatal.3c02758 · Cited by 19

Recent Advancements and Developments in the Biological Importance of 1,3,5‐Triazines

Rathod, B., Pawar, S., Puri, S., Diwan, A., & Kumar, K. (2024) · ChemistrySelect · doi:10.1002/slct.202303655 · Cited by 19

Design and Synthesis of New Biprivileged Molecular Scaffolds: Indolo‐Fused Benzodiazepinyl/quinoxalinyl benzimidazoles

Barve, I. J., Chen, C., Salunke, D. B., Chung, W., & Sun, C. (2012) · Chemistry - An Asian Journal · doi:10.1002/asia.201200121 · Cited by 19

Multicomponent, Mannich-type assembly process for generating novel, biologically-active 2-arylpiperidines and derivatives

Hardy, S., & Martin, S. F. (2014) · Tetrahedron · doi:10.1016/j.tet.2014.06.045 · Cited by 19

Amide-controlled, one-pot synthesis of tri-substituted purines generates structural diversity and analogues with trypanocidal activity

y Villatoro, M. J. P. D. L. I., Unciti-Broceta, J. D., Contreras‐Montoya, R., Garcia-Salcedo, J. A., Mezo, M. Á. G., Unciti‐Broceta, A., & Díaz‐Mochon, J. J. (2015) · Scientific Reports · doi:10.1038/srep09139 · Cited by 19

Spirocyclic amino alcohol building blocks prepared via a Prins-type cyclization in aqueous sulfuric acid

Lukin, A. Y., Bagnyukova, D., Kalinchenkova, N., Zhurilo, N., & Krasavin, M. (2016) · Tetrahedron Letters · doi:10.1016/j.tetlet.2016.06.054 · Cited by 19

A modular CuI-L-proline catalyzed one-pot route for the rapid access of constrained and privileged hetero-atom-linked medium-sized ring systems

Srinivasulu, V., Janda, K. D., Abu‐Yousef, I. A., O’Connor, M. J., & Al‐Tel, T. H. (2017) · Tetrahedron · doi:10.1016/j.tet.2017.02.061 · Cited by 19

3-Selenocyanate-indoles as new agents for the treatment of superficial and mucocutaneous infections

Quatrin, P. M., Lana, D. F. D., Bazana, L. C. G., de Oliveira, L. F. S., Teixeira, M. L., Silva, E. E., Lopes, W., Canto, R. F. S., Silveira, G. P., & Fuentefría, A. M. (2018) · New Journal of Chemistry · doi:10.1039/c8nj04935a · Cited by 20

Sulfonylation of 1,4‐Diazabicyclo[2.2.2]octane: Charge‐Transfer Complex Triggered C−N Bond Cleavage

Fu, Y. H., Xu, Q., Li, Q., Li, M., Shi, C., & Du, Z. (2019) · ChemistryOpen · doi:10.1002/open.201800251 · Cited by 19

Efficient two-step synthesis of structurally diverse indolo[2,3- b ]quinoline derivatives

Kundal, S., Chakraborty, B., Paul, K., & Jana, U. (2019) · Organic & Biomolecular Chemistry · doi:10.1039/c8ob03033b · Cited by 19

Synthesis, anti-proliferative activity, theoretical and 1H NMR experimental studies of Morita–Baylis–Hillman adducts from isatin derivatives

Brito, V. B. M., Santos, G. F., Silva, T. D. S., Souza, J. L. C., Militão, G. C. G., Martins, F. T., Silva, F. P. L., Oliveira, B. G. D., Araújo, E. C. D. C., Vasconcellos, M. L. A. A., et al. (2019) · Molecular Diversity · doi:10.1007/s11030-019-09950-7 · Cited by 19

Translating antibody-binding peptides into peptoid ligands with improved affinity and stability

Bordelon, T., Bobay, B. G., Murphy, A., Reese, H. R., Shanahan, C. C., Odeh, F., Broussard, A., Kormos, C. M., & Menegatti, S. (2019) · Journal of Chromatography A · doi:10.1016/j.chroma.2019.05.047 · Cited by 18

Synthesis of 2- and 3-Indolylpyrroles via 1,3-Dipolar Cycloadditions of Münchnones and Nitroalkenes

Gribble, G. W., & Lopchuk, J. M. (2010) · Heterocycles · doi:10.3987/com-10-s(e)125 · Cited by 19

Sc(OTf) 3 -Catalyzed Synthesis of Indoles and SnCl 4 -Mediated Regioselective Hydrochlorination of 5-(Arylamino)pent-3-yn-2-ones

Yang, F., Ji, K., Ali, S., & Liang, Y. (2011) · The Journal of Organic Chemistry · doi:10.1021/jo201514q · Cited by 19

One‐Pot Synthesis of 3‐(2‐Fluoroalkenyl)indoles

Aldoshin, A. S., Tabolin, A. A., Ioffe, S. L., & Nenajdenko, V. G. (2019) · European Journal of Organic Chemistry · doi:10.1002/ejoc.201900573 · Cited by 19

Purine-based Ir( iii ) complexes for sensing viscosity of endo-plasmic reticulum with fluorescence lifetime imaging microscopy

Liu, X., Li, K., Shi, L., Zhang, H., Liu, Y., Wang, H., Wang, N., & Yu, X. (2021) · Chemical Communications · doi:10.1039/d0cc07867k · Cited by 19

Annulation of 2‐Alkynylanilines: The Versatile Chemical Compounds

Vavsari, V. F., Nikbakht, A., & Balalaie, S. (2022) · Asian Journal of Organic Chemistry · doi:10.1002/ajoc.202100772 · Cited by 19

Stereoselective Synthesis of Polysubstituted Piperazines and Oxopiperazines. Useful Building Blocks in Medicinal Chemistry

Mordini, A., Reginato, G., Calamante, M., & Zani, L. (2014) · Current Topics in Medicinal Chemistry · doi:10.2174/1568026614666140423114013 · Cited by 19

Concise Xanthine Synthesis through a Double‐Amidination Reaction of a 6‐Chlorouracil with Amidines using Base‐Metal Catalysis

Morel, B., Franck, P., Bidange, J., Sergeyev, S. A., Smith, D. A., Moseley, J. D., & Maes, B. U. W. (2016) · ChemSusChem · doi:10.1002/cssc.201601483 · Cited by 19

“In Water”: Organocatalyzed Diastereoselective Multicomponent Reactions toward 2-Azapyrrolizidine Alkaloid Scaffolds

Rajarathinam, B., Kumaravel, K., & Vasuki, G. (2017) · ACS Combinatorial Science · doi:10.1021/acscombsci.7b00038 · Cited by 19

Minisci C–H Alkylation of Heterocycles with Unactivated Alkyl Iodides Enabled by Visible Light Photocatalysis

Yedase, G. S., Murgeshan, R., & Yatham, V. R. (2025) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.4c03151 · Cited by 18

A three-component synthesis of aryl(heteroaryl)acylamides

Loska, R., & Bukowska, P. (2015) · Organic & Biomolecular Chemistry · doi:10.1039/c5ob01355k · Cited by 18

Neurotrophe Naturstoffe – ihre Chemie und Biologie

Xu, J., Lacoske, M. H., & Theodorakis, E. A. (2013) · Angewandte Chemie · doi:10.1002/ange.201302268 · Cited by 18

DMAP-catalyzed alkylation of isatin N , N ′-cyclic azomethine imine 1,3-dipoles with Morita–Baylis–Hillman carbonates

Hu, S., Zhang, J., & Jin, Q. (2018) · New Journal of Chemistry · doi:10.1039/c8nj00234g · Cited by 18

Synthesis of Quinoline‐Thiazolidine‐2,4‐dione Coupled Pyrazoles as in vitro EGFR Targeting Anti‐Breast Cancer Agents and Their in silico Studies

Bangaru, M., Nukala, S. K., Kannekanti, P. K., Narsimha, S., Manchal, R., & Thirukovela, N. S. (2023) · ChemistrySelect · doi:10.1002/slct.202204414 · Cited by 18

Visible-Light-Induced PhI(OAc)2-Mediated Alkylation of Heteroarenes with Simple Alkanes and Ethers

Mantry, L., & Gandeepan, P. (2024) · The Journal of Organic Chemistry · doi:10.1021/acs.joc.4c00140 · Cited by 18

Design, synthesis of combretastatin A-4 piperazine derivatives as potential antitumor agents by inhibiting tubulin polymerization and inducing autophagy in HCT116 cells

Zhang, H., Li, M., Zhou, X., Tang, L., Chen, G., & Zhang, Y. (2024) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2024.116497 · Cited by 18

4-Oxo-1,4-dihydro-quinoline-3-carboxamides as BACE-1 inhibitors: Synthesis, biological evaluation and docking studies

Liu, P., Niu, Y., Wang, C., Sun, Q., Zhai, Y., Yu, J., Sun, J., Xu, F., Yan, G., Huang, W., et al. (2014) · European Journal of Medicinal Chemistry · doi:10.1016/j.ejmech.2014.04.025 · Cited by 18

Complex chromene derivatives through a silver-catalysed cascade reaction of simple o-alkynylsalicylaldehydes and alkenes

Arto, T., Fernández, P., Fañanás, F. J., & Rodríguez, F. (2016) · Chemical Communications · doi:10.1039/c6cc07801j · Cited by 18

Coupling Reactions of Alkynyl Indoles and CO 2 by Bicyclic Guanidine: Origin of Catalytic Activity?

Kee, C. W., Peh, K. Q. E., & Wong, M. W. (2017) · Chemistry - An Asian Journal · doi:10.1002/asia.201700338 · Cited by 18

Efficient Multicomponent Approach to the Medicinally Relevant 5-aryl-chromeno[2,3-b]pyridine Scaffold

Elinson, M. N., Vereshchagin, A. N., Anisina, Y. E., & Egorov, M. P. (2017) · Polycyclic aromatic compounds · doi:10.1080/10406638.2017.1363062 · Cited by 18

The cationic tetradecapeptide mastoparan as a privileged structure for drug discovery: Enhanced antimicrobial properties of mitoparan analogues modified at position-14

Howl, J., Howl, L., & Jones, S. (2018) · Peptides · doi:10.1016/j.peptides.2018.01.007 · Cited by 18

Sulfamic Acid‐Catalyzed One‐Pot Synthesis of a New Series of Biologically Relevant Indole‐Uracil Molecular Hybrids in Water at Room Temperature

Brahmachari, G., Begam, S., & Nurjamal, K. (2018) · ChemistrySelect · doi:10.1002/slct.201800488 · Cited by 18

Catalytic Dehydrative Lactonization of Allylic Alcohols

Liu, J., Miotto, R. J., Segard, J., Erb, A. M., & Aponick, A. (2018) · Organic Letters · doi:10.1021/acs.orglett.8b01063 · Cited by 18

Structural insights into pharmacophore-assistedin silicoidentification of protein–protein interaction inhibitors for inhibition of human toll-like receptor 4 – myeloid differentiation factor-2 (hTLR4−MD-2) complex

Mishra, V., & Pathak, C. (2018) · Journal of Biomolecular Structure and Dynamics · doi:10.1080/07391102.2018.1474804 · Cited by 18

1,4-Benzodioxane Lignans: An Efficient, Asymmetric Synthesis of Flavonolignans and Study of Neolignan Cytotoxicity and Antiviral Profiles

Pilkington, L. I., Wagoner, J., Kline, T. B., Polyak, S. J., & Barker, D. L. A. (2018) · Journal of Natural Products · doi:10.1021/acs.jnatprod.8b00416 · Cited by 18

Metal-, photocatalyst-, and light-free late-stage C–H alkylation of N-heteroarenes with organotrimethylsilanes using persulfate as a stoichiometric oxidant

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