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Crystal Structure of the Intrinsically Flexible Addiction Antidote MazE

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The Effect of pH on β2 Adrenoceptor Function

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Subcellular Organization of GPCR Signaling

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GPCR signaling along the endocytic pathway

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Neuropeptides and Neuropeptide Receptors: Drug Targets, and Peptide and Non‐Peptide Ligands: a Tribute to Prof.Dieter Seebach

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GPCR-targeting nanobodies: attractive research tools, diagnostics, and therapeutics

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Covalent agonists for studying G protein-coupled receptor activation

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Fragment Screening at Adenosine-A3 Receptors in Living Cells Using a Fluorescence-Based Binding Assay

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Diversity and functional properties of bistable pigments

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Allosteric nanobodies uncover a role of hippocampal mGlu2 receptor homodimers in contextual fear consolidation

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Nanobodies to study protein conformational states

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Comparing Class A GPCRs to bitter taste receptors

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Conformational plasticity of ligand-bound and ternary GPCR complexes studied by 19F NMR of the β1-adrenergic receptor

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Conformationally selective RNA aptamers allosterically modulate the β2-adrenoceptor

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How Can Mutations Thermostabilize G-Protein-Coupled Receptors?

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Breaking the barriers in membrane protein crystallography

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Large-scale production and protein engineering of G protein-coupled receptors for structural studies

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A conserved molecular switch in Class F receptors regulates receptor activation and pathway selection

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New concepts and aids to facilitate crystallization

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New Technologies for Elucidating Opioid Receptor Function

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Aminergic GPCR–Ligand Interactions: A Chemical and Structural Map of Receptor Mutation Data

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Structurally Enabled Discovery of Adenosine A 2A Receptor Antagonists

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Active state structures of G protein-coupled receptors highlight the similarities and differences in the G protein and arrestin coupling interfaces

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Isolation of state-dependent monoclonal antibodies against the 12-transmembrane domain glucose transporter 4 using virus-like particles

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Location Bias as Emerging Paradigm in GPCR Biology and Drug Discovery

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Structure‐Based Discovery of Allosteric Modulators of Two Related Class B G‐Protein‐Coupled Receptors

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Functional selectivity of GPCR signaling in animals

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Antibodies and protein misfolding: From structural research tools to therapeutic strategies

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Structural changes in the transport cycle of the mitochondrial ADP/ATP carrier

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A general approach for stabilizing nanobodies for intracellular expression

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Nanobodies Based on a Sandwich Immunoassay for the Detection of Staphylococcal Enterotoxin B Free from Interference by Protein A

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The fine art of integral membrane protein crystallisation

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Molecular Basis of Opioid Action: From Structures to New Leads

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Use of transmission electron microscopy to identify nanocrystals of challenging protein targets

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Nanobodies detecting and modulating GPCRs outside in and inside out

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Enabling STD-NMR fragment screening using stabilized native GPCR: A case study of adenosine receptor

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Structure of cyclin G-associated kinase (GAK) trapped in different conformations using nanobodies

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Receptor signals come in waves

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The G‐Protein‐Coupled Neuropeptide Y Receptor Type 2 is Highly Dynamic in Lipid Membranes as Revealed by Solid‐State NMR Spectroscopy

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Proof of dual-topology architecture of Fluc F− channels with monobody blockers

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G protein-coupled receptors in rheumatology

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Heterologous desensitization of cardiac β-adrenergic signal via hormone-induced βAR/arrestin/PDE4 complexes

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A Molecular Pharmacologist’s Guide to G Protein–Coupled Receptor Crystallography

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Computational and Experimental Analysis of the Transmembrane Domain 4/5 Dimerization Interface of the Serotonin 5-HT1A Receptor

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Protein crystallization: Eluding the bottleneck of X-ray crystallography

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Endomembrane-Based Signaling by GPCRs and G-Proteins

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Advances in NMR structures of integral membrane proteins

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Neutralization of Human Interleukin 23 by Multivalent Nanobodies Explained by the Structure of Cytokine–Nanobody Complex

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AAV‐mediated delivery of an anti‐BACE1 VHH alleviates pathology in an Alzheimer's disease model

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Biasing GPCR Signaling from Inside

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Generation, characterization and structural data of chymase binding proteins based on the human Fyn kinase SH3 domain

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Chemical Biology Methods for Investigating G Protein-Coupled Receptor Signaling

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Site-Specific Epitope Tagging of G Protein-Coupled Receptors by Bioorthogonal Modification of a Genetically Encoded Unnatural Amino Acid

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Crystal structure of a LacY–nanobody complex in a periplasmic-open conformation

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Identification and characterization of Nanobodies targeting the EphA4 receptor

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Complex Formation between VEGFR2 and the β2-Adrenoceptor

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A cDNA Immunization Strategy to Generate Nanobodies against Membrane Proteins in Native Conformation

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Nanobody-Based Biologics for Modulating Purinergic Signaling in Inflammation and Immunity

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Transmission electron microscopy for the evaluation and optimization of crystal growth

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Metadynamics simulations of ligand binding to GPCRs

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Directed evolution of nanobody chaperones that stabilize GPCR:G‐protein complexes

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Extracellular Nanobody Screening using Conformationally Stable GPCRPreprint

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Nanobodies to Study G Protein–Coupled Receptor Structure and Function

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G-Protein Peptidomimetics Stabilize GPCR Active State Conformations

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Nanobody stabilization of G protein–coupled receptors (GPCRs) for activated structure determination

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