Modulators of Protein–Protein Interactions
Milroy, Lech-Gustav, Grossmann, Tom N., Hennig, Sven, Brunsveld, Luc, Ottmann, Christian·2014·Chemical Reviews
Cited by (523)
Items 301–400 of 523
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- A systematic approach to identify host targets and rapidly deliver broad-spectrum antiviralsJulien Olivet, Sibusiso B. Maseko, Alexander N. Volkov, Kourosh Salehi‐Ashtiani, Kalyan Das, Michael A. Calderwood, Jean‐Claude Twizere, Christoph Gorgulla · 2022 · Molecular Therapy
- New Compound Classes: Protein–Protein InteractionsChristian Ottmann · 2015 · Handbook of experimental pharmacology
- Electrostatic roles in electron transfer from [NiFe] hydrogenase to cytochrome c 3 from Desulfovibrio vulgaris Miyazaki FYu Sugimoto, Yuki Kitazumi, Osamu Shirai, Koji Nishikawa, Yoshiki Higuchi, Masahiro Yamamoto, Kenji Kano · 2017 · Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics
- HBx-Derived Constrained Peptides Inhibit the Secretion of Hepatitis B Virus AntigensXiaodan Cai, Weihao Zheng, Xiaodong Shi, Longjian Chen, Zhihong Liu, Zigang Li · 2018 · Molecular Pharmaceutics
- Lipidated Stapled Peptides Targeting the Acyl Binding Protein UNC119Philipp M. Cromm, Hélène Adihou, Shobhna Kapoor, Mercedes Vázquez–Chantada, Paul R. J. Davey, David Longmire, Elisabeth Hennes, Walter Hofer, Philipp Küchler, Elisabetta Chiarparin et al. · 2019 · ChemBioChem
- A new insight into subinteractomes of functional antagonists: Thromboxane (CYP5A1) and prostacyclin (CYP8A1) synthasesPavel V. Ershov, Evgeniy O. Yablokov, Victor Gavrilovich Zgoda, Yuri V. Mezentsev, Oksana V. Gnedenko, Leonid A. Kaluzhskiy, Andrey V. Svirid, Andrei A. Gilep, Sergey A. Usanov, Alexis S. Ivanov · 2021 · Cell Biology International
- Recent developments in the utility of saturated azaheterocycles in peptidomimeticsManish K. Singh, Mahesh K. Lakshman · 2021 · Organic & Biomolecular Chemistry
- Fragment‐Based Stabilizers of Protein–Protein Interactions through Imine‐Based TetheringM. Wolter, Dario Valenti, Peter J. Cossar, Laura M. Levy, Stanimira Hristeva, Thorsten Genski, Torsten Hoffmann, Luc Brunsveld, Dimitrios Tzalis, Christian Ottmann · 2020 · Angewandte Chemie
- A Chemical Inhibitor of the Skp2/p300 Interaction that Promotes p53‐Mediated ApoptosisMisook Oh, Ji Hoon Lee, Heejo Moon, Yu-Jung Hyun, Hyun‐Suk Lim · 2015 · Angewandte Chemie
- Dual Functional Modification of Alkaline Amino Acids Induces the Self‐Assembly of Cylinder‐Like Tobacco Mosaic Virus Coat Proteins into Gear‐Like ArchitecturesJian‐Ting Zhang, Ranjith Kumar Kankala, Yihao Zhou, Jinchen Dong, Ai‐Zheng Chen, Qiangbin Wang · 2019 · Small
- Exploring Framework Nucleic Acids: A Perspective on Their Cellular ApplicationsZhaoyang Wang, Xin Wang, Yao He, Hui Chen Wu, Rui Mao, Haiyuan Wang, Liping Qiu · 2024 · JACS Au
- Harnessing Allostery to Modulate Protein–Protein Interactions: From Function to Therapeutic InnovationsSutanu Mukhopadhyay, Krishnendu Sinha, Suman Chakrabarty · 2025 · Journal of Molecular Biology
- Direkte Modulation von Aktivität und Funktion kleiner GTPasenPhilipp M. Cromm, Jochen Spiegel, Tom N. Grossmann, Herbert Waldmann · 2015 · Angewandte Chemie
- Design criteria for minimalist mimics of protein–protein interface segmentsJaru Taechalertpaisarn, Rui-Liang Lyu, Maritess Arancillo, Chen‐Ming Lin, Zhengyang Jiang, Lisa M. Pérez, Thomas R. Ioerger, Kevin Burgess · 2018 · Organic & Biomolecular Chemistry
- Different phosphorylation and farnesylation patterns tune Rnd3–14-3-3 interaction in distinct mechanismsJun Hu, Xue-Meng Sun, Jingyun Su, Yufen Zhao, Yong‐Xiang Chen · 2021 · Chemical Science
- When Supramolecular Chemistry Meets Chemical Biology: New Strategies to Target Proteins through Host‐Guest InteractionsWenbing Cao, Xuewen Qin, Tao Liu · 2021 · ChemBioChem
- Coacervate Formed by an ATP-Binding Aptamer and Its Dynamic Behavior under Nonequilibrium ConditionsZhijun Liu, Jiaxin Chen, Qingwen Bai, Ya-nan Lin, Dehai Liang · 2022 · Langmuir
- Discovery of 14‐3‐3 PPI Stabilizers by Extension of an Amidine‐Substituted Thiophene FragmentQi Wu, Federica Centorrino, X. Guillory, M. Wolter, Christian Ottmann, Peter J. Cossar, Luc Brunsveld · 2023 · ChemBioChem
- Synthesis of a Bcl9 Alpha-Helix Mimetic for Inhibition of PPIs by a Combination of Electrooxidative Phenol Coupling and Pd-Catalyzed Cross CouplingMartin Vareka, Benedikt Dahms, Mario Lang, Minh Hao Hoang, Melanie Trobe, Hansjörg Weber, Maximilian M. Hielscher, Siegfried R. Waldvogel, Rolf Breinbauer · 2020 · Catalysts
- Allosteric ModulatorsShaoyong Lu, Jinyan Zhang · 2016 · Elsevier eBooks
- Terminal protection of peptides by interactions with proteins: A “signal-on” peptide-templated gold nanocluster beacon for label-free protein detectionQian Wen, Sili Yi, Qinlu Lin, Li‐Juan Tang, Jian‐Hui Jiang · 2021 · Talanta
- Bispidine as a β-strand nucleator: from a β-arch to self-assembled cages and vesiclesHanuman Singh, Akshay Chenna, Upanshu Gangwar, Julie Borah, Gaurav Goel, V. Haridas · 2021 · Chemical Science
- A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 5: A Complete Set of Pyridine Boronic Acid Pinacol Esters Featuring Side Chains of Proteinogenic Amino AcidsMelanie Trobe, Till Schreiner, Martin Vareka, Sebastian Grimm, Bernhard Wölfl, Rolf Breinbauer · 2022 · European Journal of Organic Chemistry
- Chemical synthesis of a reported p47phox/p22phox inhibitor and characterization of its instability and irreproducible activityJie Zang, Yves Cambet, Vincent Jaquet, Anders Bach · 2023 · Frontiers in Pharmacology
- Straightforward model construction and analysis of multicomponent biomolecular systems in equilibriumNick H. J. Geertjens, Pim J. de Vink, Tim Wezeman, Albert Jan Markvoort, Luc Brunsveld · 2023 · RSC Chemical Biology
- Recent advances in the modulation of amyloid protein aggregation using the supramolecular host-guest approachesDebabrata Maity · 2023 · Biophysical Chemistry
- Disulfide Click Reaction for Stapling of S‐terminal PeptidesQing Yu, Leiyang Bai, Xuefeng Jiang · 2023 · Angewandte Chemie
- Assembly and Functionality of 2D Protein ArraysMingming Du, Fanmeng Zeng, YueFei Wang, Yongjun Li, Guangcun Chen, Jiang Jiang, Qiangbin Wang · 2025 · Advanced Science
- Site-selective modification of native proteinsYujun Kim, Han Yi, Kyungdeok Seo, Hyun Soo Lee, Injae Shin · 2025 · Trends in Chemistry
- TAX1BP3 Is a SUMOylated Nucleocytoplasmic Shuttling Protein and Protects Against Vascular Neointimal HyperplasiaHanyan Yang, Yulong Zhong, Wenjie Guo, Wenjing Guo, Boliang Chen, Zexuan Lin, Qin Zhang, Rongjun Zou, Xiaolong Cao, Fengxian Li et al. · 2025 · Circulation
- Stalis: A Computational Method for Template‐Based Ab Initio Ligand DesignHui Sun Lee, Wonpil Im · 2019 · Journal of Computational Chemistry
- Bicyclic Schellman Loop Mimics (BSMs): Rigid Synthetic C-Caps for Enforcing Peptide HelicityTianxiong Mi, Duyen Nguyen, Kevin Burgess · 2023 · ACS Central Science
- Bivalent molecular mimicry by ADP protects metal redox state and promotes coenzyme B 12 repairHarsha Gouda, Romila Mascarenhas, Markus Ruetz, Madeline Yaw, Ruma V. Banerjee · 2023 · Proceedings of the National Academy of Sciences
- Molecular electrostatic potential and volume-aided drug design based on the isoindolinone-containing cyclopeptide S-PK6Lei Zhao, Tingting Li, Hongyu Xu, Xiong Zhang, Huiming Lin, Na Liu, Yingxue Jin, Zhiqiang Wang · 2023 · New Journal of Chemistry
- Facile Peptide Macrocyclization and Multifunctionalization via Cyclen InstallationTsz‐Lam Cheung, Leo K. B. Tam, Wing‐Sze Tam, Leilei Zhang, Hei‐Yui Kai, Waygen Thor, Yue Wu, Pak‐Lun Lam, Yik‐Hoi Yeung, Chen Xie et al. · 2024 · Small Methods
- Novel peptide—based inhibitor for targeted inhibition of T cell functionAshna Gauthaman, Rini Jacob, Sneha Pasupati, Rajadurai Abarna, C. George Priya Doss, Anbalagan Moorthy · 2021 · Journal of Cell Communication and Signaling
- A Non‐coded β2,2‐Amino Acid with Isoxazoline Core Able to Stabilize Peptides Folding through an Unprecedented Hydrogen BondRaffaella Bucci, Francesco Vaghi, Davide Di Lorenzo, Francesco Anastasi, Gianluigi Broggini, Leonardo Lo Presti, Alessandro Contini, Maria Luisa Gelmi · 2022 · European Journal of Organic Chemistry
- Explaining RANKL inhibition by OPG through quantum biochemistry computations and insights into peptide-design for the treatment of osteoporosisBruno Lopes de Sousa, Ito L. Barroso-Neto, Evanildo F. Oliveira, Emerson Alberto Fonseca, Pedro de Lima‐Neto, Luiz O. Ladeira, V. N. Freire · 2016 · RSC Advances
- A Novel Long‐Range n to π* Interaction Secures the Smallest known α‐Helix in WaterHuy N. Hoang, Chongyang Wu, Timothy A. Hill, Aline D. de Araujo, Paul V. Bernhardt, Ligong Liu, David P. Fairlie · 2019 · Angewandte Chemie
- Small-molecule inhibitors of the CD40–CD40L costimulatory interaction are effective in pancreatic islet transplantation and prevention of type 1 diabetes modelsSung-Ting Chuang, Oscar Alcazar, B.M. Watts, Midhat H. Abdulreda, Péter Buchwald · 2024 · Frontiers in Immunology
- Integrating Protein Interaction Surface Prediction with a Fragment-Based Drug Design: Automatic Design of New Leads with Fragments on Energy SurfacesLuca Torielli, Stefano Artin Serapian, Lara Mussolin, Elisabetta Moroni, Giorgio Colombo · 2022 · Journal of Chemical Information and Modeling
- The role of N-terminal proline in stabilizing the Ant–Pro zipper motifSanjeev Kheria, Roshna V. Nair, Amol S. Kotmale, Pattuparambil Ramanpillai Rajamohanan, Gangadhar J. Sanjayan · 2015 · New Journal of Chemistry
- Light-driven release of cucurbit[8]uril from a bivalent cagePim J. de Vink, Tim van der Hek, Luc Brunsveld · 2021 · Chemical Science
- Recent Advances in β-catenin/BCL9 protein–protein Interaction InhibitorsHao Zhang, Ya Bao, Chenglong Liu, Jianqi Li, Di Zhu, Qingwei Zhang · 2021 · Future Medicinal Chemistry
- Head-to-Tail Cross-Linking to Generate Bicyclic Helical Peptides with Enhanced Helicity and Proteolytic StabilityKai Chen, Yang Tang, Meng Yao Wu, Xiao-Cui Wan, Yanni Zhang, Xiaoxu Chen, Fei-Qiang Yu, Zhihui Cui, Jinming Ma, Zhaocai Zhou et al. · 2021 · Organic Letters
- On-Resin Synthesis of Linear Aryl Thioether Containing Peptides and in-Solution Cyclization via Cysteine SNAr ReactionJian Li, Weihong Lai, Ao Pang, Lu Liu, Lianbao Ye, Xiao‐Feng Xiong · 2022 · Organic Letters
- Binding Dynamics of a Stapled Peptide Targeting the Transcription Factor NF−YCanan Durukan, Federica Arbore, Rasmus Klintrot, Carlo Bigiotti, Ioana Mariuca Ilie, Jocelyne Vreede, Tom N. Grossmann, Sven Hennig · 2024 · ChemBioChem
- Probing Protein Surfaces: QSAR Analysis with Helix MimeticsValeria Azzarito, Philip R. Rowell, Anna Barnard, Thomas A. Edwards, Andrew Macdonald, Stuart L. Warriner, Andrew John Wilson · 2015 · ChemBioChem
- Cucurbit[8]uril Reactivation of an Inactivated Caspase‐8 Mutant Reveals Differentiated Enzymatic Substrate ProcessingDung T. Dang, Arthur H. A. M. van Onzen, Yvonne L. Dorland, Luc Brunsveld · 2018 · ChemBioChem
- Peptidomimetics IIWilliam D. Lubell · 2016 · Topics in heterocyclic chemistry
- From Degraders to Molecular Glues: New Ways of Breaking Down Disease‐Associated ProteinsYvonne A. Nagel, Adrian Britschgi, Antonio Ricci · 2021 · Wiley eBooks
- Molecular Glue Degraders: From Serendipity to Hunting and DesignLuis Nieto‐Barrado, Ana Domostegui, Cristina Mayor‐Ruiz · 2022 · Wiley eBooks
- Patenting perspective on Keap1 inhibitors (2019–2024)Yongfu Luo, Wenlong Yang, Yuan Zhang, Shutong Jiang, Jingyu Zhu, Xiangyang Li, Qidong You, Mengchen Lu · 2025 · Expert Opinion on Therapeutic Patents
- Interrogating the potential of helical aromatic foldamers for protein recognitionSunbum Kwon, Vasily Morozov, Lingfei Wang, Pradeep K. Mandal, Stéphane Chaignepain, Céline Douat, Ivan Huc · 2024 · Organic & Biomolecular Chemistry
- ATP Inhibits the Transcription Factor STAT5bAngela Berg, Bianca Sperl, Thorsten Berg · 2019 · ChemBioChem
- Solid-phase parallel synthesis of 1,3-thiazole library adorned with dipeptidyl chainsMin-Jeong Cha, Aizhan Abdildinova, Young‐Dae Gong · 2020 · Tetrahedron
- Protein-protein interaction and interference of carcinogenesis by supramolecular modificationsOluwatosin A. Saibu, Opeyemi Sodiq Hammed, Oladapo O. Oladipo, Tope Tunji Odunitan, Temitope M. Ajayi, Aderonke J. Adejuyigbe, Boluwatife T. Apanisile, Oluwatoba Emmanuel Oyeneyin, Adenrele T. Oluwafemi, Tolulope Ayoola et al. · 2023 · Bioorganic & Medicinal Chemistry
- Deciphering key genes involved in cisplatin resistance in kidney renal clear cell carcinoma through a combined in silico and in vitro approachMuneeba Malik, MAMOONA MAQBOOL, TOOBA NISAR, TAZEEM AKHTER, Javed Ahmed Ujan, Alanood Saeed Algarni, Fakhria A. Al‐Joufi, SULTAN SHAFI K. ALANAZI, MOHAMMAD HADI ALMOTARED, Mounir Mohamed Salem-Bekhit et al. · 2023 · Oncology Research Featuring Preclinical and Clinical Cancer Therapeutics
- Bisphosphonate ligand mediated ultrasensitive capacitive protein sensor: complementary match of supramolecular and dynamic chemistryGizem Ertürk, Maedeh Akhoundian, Kyra Lueg-Althoff, Sudhirkumar Shinde, Sing Yee Yeung, Martin Hedström, Thomas H. Schrader, Bo Mattìasson, Börje Sellergren · 2018 · New Journal of Chemistry
- Helix-Constrained Peptides Constructed by Head-to-Side Chain Cross-Linking StrategiesXiaoxu Chen, Yang Tang, Meng Yao Wu, Yanni Zhang, Kai Chen, Zhaocai Zhou, Ge‐Min Fang · 2021 · Organic Letters
- HOPPI-NMR: Hot-Peptide-Based Screening Assay for Inhibitors of Protein–Protein Interactions by NMRDiego Brancaccio, Salvatore Di Maro, Linda Cerofolini, Stefano Giuntini, Marco Fragai, Claudio Luchinat, Stefano Tomassi, Antonio Limatola, Pasquale Russomanno, Francesco Merlino et al. · 2020 · ACS Medicinal Chemistry Letters
- A NanoBRET-based assay monitoring interactions in the USP18 signaling hub identifies the first cell-penetrant small molecule compromising USP18/ISG15 bindingSandra Hess, Marta Campos Alonso, Michael J. D. Brand, Susan Lauw, Urs Lindenmann, Katharina Göbel, Paul P. Geurink, Günter Fritz, Rainer Riedl, Klaus‐Peter Knobeloch · 2025 · bioRxiv (Cold Spring Harbor Laboratory)
- De Novo Discovery of α,α-Disubstituted α-amino Acid-Containing α-helical Peptides as Competitive PPARγ PPI InhibitorsMaxwell Sigal, Markus Egner, Chikako Okada, Daniel Merk, Toru Sengoku, Takayuki Katoh, Hiroaki Suga · 2025 · Journal of the American Chemical Society
- Computational model predicts protein binding sites of a luminescent ligand equipped with guanidiniocarbonyl-pyrrole groupsNeda Rafieiolhosseini, Matthias Killa, Thorben Neumann, Niklas Tötsch, Jean‐Noël Grad, Alexander Höing, Thies Dirksmeyer, Jochen Niemeyer, Christian Ottmann, Shirley K. Knauer et al. · 2022 · Beilstein Journal of Organic Chemistry
- Multivalent Molecular Tweezers Disrupt the Essential NDC80 Interaction with MicrotubulesJonas Neblik, Abbna Kirupakaran, Christine Beuck, Joel Mieres‐Pérez, Felix C. Niemeyer, My‐Hue Le, Ursula Telgheder, Jessica Felice Schmuck, Alexander Dudziak, Peter Bayer et al. · 2023 · Journal of the American Chemical Society
- Machine learning of metabolite–protein interactions from model-derived metabolic phenotypesMahdis Habibpour, Zahra Razaghi‐Moghadam, Zoran Nikoloski · 2024 · NAR Genomics and Bioinformatics
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- Towards optimizing peptide-based inhibitors of protein–protein interactions: predictive saturation variation scanning (PreSaVS)Kristina Hetherington, Som Dutt, Amaurys Ávila Ibarra, Emma E. Cawood, Fruzsina Hóbor, Derek N. Woolfson, Thomas A. Edwards, Adam S. Nelson, Richard Barry Sessions, Andrew John Wilson · 2021 · RSC Chemical Biology
- Inhibition of Protein–Protein Interactions: New Options for Developing Drugs against Neglected Tropical DiseasesThorsten Berg · 2017 · Angewandte Chemie International Edition
- Synthesis of Bis-Glyoxylamide Peptidomimetics Derived from Bis-N-acetylisatins Linked at C5 by a Methylene or Oxygen BridgeVenty Suryanti, Ruonan Zhang, Vina R. Aldilla, Mohan Madhav Bhadbhade, Naresh Kumar, David StC. Black · 2019 · Molecules
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- Supramolecular self-assembly: A facile way to fabricate protein and peptide nanomaterialsLuyang Zhao, Xuehai Yan · 2020 · Elsevier eBooks
- A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 3: Iodophenyltriflate Core Fragments Featuring Side Chains of Proteinogenic Amino AcidsMelanie Trobe, Martin Vareka, Till Schreiner, Patrick Simon Dobrounig, Carina Doler, Ella B. Holzinger, Andreas Steinegger, Rolf Breinbauer · 2022 · European Journal of Organic Chemistry
- Rationally Designed Semisynthetic Natural Product Analogues for Stabilization of 14‐3‐3 Protein–Protein InteractionsSebastian A. Andrei, Pim J. de Vink, Eline Sijbesma, Ling Han, Luc Brunsveld, Nobuo Kato, Christian Ottmann, Yusuke Higuchi · 2018 · Angewandte Chemie
- Bicyclic β‐Sheet Mimetics that Target the Transcriptional Coactivator β‐Catenin and Inhibit Wnt SignalingMathias Wendt, Rosa Bellavita, Alan Gerber, Nina‐Louisa Efrém, Thirza van Ramshorst, Nicholas M. Pearce, Paul R. J. Davey, Isabel Everard, Mercedes Vázquez–Chantada, Elisabetta Chiarparin et al. · 2021 · Angewandte Chemie
- Analysis of the interaction of cyclosporine congeners with cell membrane modelsMizuka Nakao, Yuki Takechi‐Haraya, Takashi Ohgita, Hiroyuki Saito, Yosuke Demizu, Ken‐ichi Izutsu, Kumiko Sakai‐Kato · 2022 · Journal of Pharmaceutical and Biomedical Analysis
- How Do Molecular Tweezers Bind to Proteins? Lessons from X-ray CrystallographyArthur T. Porfetye, Patricia Stege, Rocio Rebollido-Rios, Daniel E. Hoffmann, Thomas H. Schrader, Ingrid R. Vetter · 2024 · Molecules
- Protein–Protein Interface Topology as a Predictor of Secondary Structure and Molecular Function Using Convolutional Deep LearningBenjamin Bouvier · 2021 · Journal of Chemical Information and Modeling
- Protein-Protein Interactions: An OverviewEdson Luiz Folador, Sandeep Tiwari, Camila E. Da Paz Barbosa, Syed Babar Jamal, Marco Da Costa Schulze, Debmalya Barh, Vasco Azevedo · 2018 · Elsevier eBooks
- SAR by 1D NMRNeal Joseph Zondlo · 2019 · Journal of Medicinal Chemistry
- Structure-based design of an aromatic helical foldamer–protein interfaceLingfei Wang, Céline Douat, Johannes Sigl, Post Sai Reddy, Lucile Fischer, Béatrice Langlois d’Estaintot, Zhiwei Liu, Vojislava Pophristic, Yuwei Yang, Yingkai Zhang et al. · 2025 · Chemical Science
- Multimodal Contrastive Learning for Protein–Protein Interaction Inhibitor PredictionZitong Zhang, Zhixian Wang, Lingling Zhao, Junjie Wang, Chunyu Wang · 2024 · IEEE International Conference on Bioinformatics and Biomedicine (BIBM)
- A pharmacological modality to sequester homomeric proteinsElla Livnah, Ohad Suss, Adi Rogel, Atar Gilat, Yuval Abdan, José A. Villegas, Ronen Gabizon, Almog Nadir, Yoav Shamir, Noam Y. Steinman et al. · 2026 · Nature Chemical Biology
- Short Oligourea Foldamers as N‐ or C‐Caps for Promoting α‐Helix Formation in WaterLaura Mauran, Coralie Assailly, Sébastien R. Goudreau, Benoı̂t Odaert, Gilles Guichard, Morgane Pasco · 2024 · ChemBioChem
- Tyrosinase‐Catalyzed Peptide Stapling Using Para‐Amino Phenylalanine and Tyrosine Anchoring ResiduesNan Wang, Zhengyang Xu, Huaxing Shen, Wei Cong, Shuai Zhang, Honggang Hu, Xiang Li · 2025 · Angewandte Chemie
- Funktionelle Inhibition der krebsrelevanten Interaktion von Survivin und Histon H3 mit einem Guanidiniumcarbonylpyrrol‐LigandenCecilia Vallet, Dennis Aschmann, Christine Beuck, Matthias Killa, Annika Meiners, Marcel Mertel, Martin Ehlers, Peter Bayer, Carsten Schmuck, Michael Giese et al. · 2020 · Angewandte Chemie
- Traceless solid-phase synthesis and β-turn propensity of 1,3-thiazole-based peptidomimeticsAizhan Abdildinova, Young‐Dae Gong · 2021 · RSC Advances
- Diazaborine-Mediated Bicyclization of Native Peptides with Inducible ReversibilityRahi M. Reja, Brittney Chau, Jianmin Gao · 2023 · Organic Letters
- Visualized and Quantitative Conformational Analysis of PeptidomimeticsHajime Takashima, Atsushi Yoshimori, Eiji Honda, Tomonori Taguri, Jun Ozawa, Masaji Kasai, Satoshi Shuto, Dai Takehara · 2021 · ACS Omega
- A Modular Synthesis of Teraryl‐Based α‐Helix Mimetics, Part 4: Core Fragments with Two Halide Leaving Groups Featuring Side Chains of Proteinogenic Amino AcidsMelanie Trobe, Julia Blesl, Martin Vareka, Till Schreiner, Rolf Breinbauer · 2022 · European Journal of Organic Chemistry
- Stackabilization: self-assembling bispidinophanesSakshi Sharma, M. V. S. Gopalakrishna, Paloth Venugopalan, Cherumuttathu Hariharan Suresh, V. Haridas · 2015 · Tetrahedron
- Modeling and Design of Peptidomimetics to Modulate Protein–Protein InteractionsAndrew M. Watkins, Richard Bonneau, Paramjit S. Arora · 2017 · Methods in molecular biology
- Mapping molecular binding by means of conformational dynamics measurementsNoelle M. do Nascimento, Augusto Juste-Dolz, Paulo R. Bueno, Isidro S. Monzó, Roberto Tejero, José Luis López-Paz, Ángel Maquieira, Sergi Morais, David Giménez-Romero · 2018 · RSC Advances
- Manumycin Polyketides Act as Molecular Glues Between UBR7 and P53 to Impair Breast Cancer PathogenicityYosuke Isobe, Mikiko Okumura, Ross White, Lynn M. McGregor, Jeffrey M. McKenna, John A. Tallarico, Markus Schirle, Thomas J. Maimone, Daniel K. Nomura · 2019 · bioRxiv (Cold Spring Harbor Laboratory)
- PPIscout: Protein–protein interaction site hotspot mapping using mixed amino acid–water molecular dynamics simulationSutanu Mukhopadhyay, Suman Chakrabarty · 2025 · Journal of Chemical Sciences
- Targeting protein protein interactions and their modulators to enable new therapeutic strategies for human diseasesAftab Alam, Maria J. Fernández-Cabezudo, Rifat Hamoudi, Basel K. al-Ramadi · 2026 · npj Systems Biology and Applications
- Advancing protein engineering via organic chemistryRaj V. Nithun, Manjeet Singh, Adam Baransi, Muhammad Jbara · 2026 · Communications Chemistry
- Examination of the Effect of N‐terminal Diproline and Charged Side Chains on the Stabilization of Helical Conformation in Alanine–based Short Peptides: A Molecular Dynamics StudyBhupesh Goyal, Kinshuk Raj Srivastava, Susheel Durani · 2016 · ChemistrySelect
- A Ligase‐Based Two‐Step Approach for the Generation of Bicyclic Peptides Containing a Benzylphenyl Thioether FrameworkHua Zhang, Hui‐Min Wei, Jun‐Hao Xue, Zhe‐Min Xia, Feng‐Hao Zheng, Xiao‐Cui Wan, Zhou Li, Ge‐Min Fang · 2025 · ChemBioChem