Modulators of Protein–Protein Interactions

Milroy, Lech-Gustav, Grossmann, Tom N., Hennig, Sven, Brunsveld, Luc, Ottmann, Christian·2014·Chemical Reviews
DOI 10.1021/cr400698c

Cited by (523)

Items 501–523 of 523

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  3. BindingDB Entry 7787: Perfluoro-tert-butyl Homoserine Is a Helix-Promoting, Highly Fluorinated, NMR-Sensitive Aliphatic Amino Acid: Detection of the Estrogen Receptor·Coactivator Protein-Protein Interaction by (19)F NMR.
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  5. BindingDB Entry 50000193: Structural Basis of Inhibition of ERα-Coactivator Interaction by High-Affinity N-Terminus Isoaspartic Acid Tethered Helical Peptides.
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  6. BindingDB Entry 50045446: Structural development of stapled short helical peptides as vitamin D receptor (VDR)-coactivator interaction inhibitors.
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  7. BindingDB Entry 50018346: Computational methods-guided design of modulators targeting protein-protein interactions (PPIs).
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  8. BindingDB Entry 50000314: Structure-Based Design of Non-natural Macrocyclic Peptides That Inhibit Protein-Protein Interactions.
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  9. BindingDB Entry 50006626: Optimization and bioevaluation of Cdc37-derived peptides: An insight into Hsp90-Cdc37 protein-protein interaction modulators.
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  10. BindingDB Entry 50001501: Structure-based virtual screening and optimization of modulators targeting Hsp90-Cdc37 interaction.
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  11. BindingDB Entry 50047509: Natural Products as Sources of New Drugs from 1981 to 2014.
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  12. BindingDB Entry 50048927: An in-tether sulfoxide chiral center influences the biophysical properties of the N-capped peptides.
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  13. BindingDB Entry 50049115: Rational design and synthesis of 1,5-disubstituted tetrazoles as potent inhibitors of the MDM2-p53 interaction.
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  14. BindingDB Entry 50008428: A Comparative Assessment Study of Known Small-Molecule Keap1-Nrf2 Protein-Protein Interaction Inhibitors: Chemical Synthesis, Binding Properties, and Cellular Activity.
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  15. BindingDB Entry 50018571: A Comprehensive Overview of Small-Molecule Androgen Receptor Degraders: Recent Progress and Future Perspectives.
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  16. BindingDB Entry 6990: Phosphorylation of Capsaicinoid Derivatives Provides Highly Potent and Selective Inhibitors of the Transcription Factor STAT5b.
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  17. BindingDB Entry 50010648: HOPPI-NMR: Hot-Peptide-Based Screening Assay for Inhibitors of Protein-Protein Interactions by NMR.
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  18. BindingDB Entry 50002786: Recent advances in peptidomimetics antagonists targeting estrogen receptor α-coactivator interaction in cancer therapy.
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  19. BindingDB Entry 50047995: Discovery and Development of Kelch-like ECH-Associated Protein 1. Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction Inhibitors: Achievements, Challenges, and Future Directions.
    BindingDB · 2018 · UC San Diego
  20. BindingDB Entry 50000979: 1,4,5-Trisubstituted Imidazole-Based p53-MDM2/MDMX Antagonists with Aliphatic Linkers for Conjugation with Biological Carriers.
    BindingDB · 2020 · UC San Diego
  21. BindingDB Entry 50008262: Recent advances in class IIa histone deacetylases research.
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  22. BindingDB Entry 50006478: Medicinal Chemistry Approaches to Heart Regeneration.
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  23. BindingDB Entry 50002721: Modulators of 14-3-3 Protein-Protein Interactions.
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