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Saquinavir Inhibits the Malaria Parasite's Chloroquine Resistance Transporter

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Synthesis and antifilarial evaluation of N1,N n- xylofuranosylated diaminoalkanes

Tiwari, V. K., Tewari, N., Katiyar, D., Tripathi, R. P., Arora, K., Gupta, S., Ahmad, R., Srivastava, A. K., Khan, M. A., Murthy, P. K., et al. (2003) · Bioorganic & Medicinal Chemistry · doi:10.1016/s0968-0896(03)00033-6 · Cited by 27 · see citing works

New approaches in vaccine development for parasitic infections

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Preparation and antimalarial activity of a novel class of carbohydrate-derived, fused thiochromans

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Targeting Ouabain- and Adducin-dependent mechanisms of hypertension and cardiovascular remodeling as a novel pharmacological approach

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Novel macrocyclic C-aryl glucoside SGLT2 inhibitors as potential antidiabetic agents

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Carbohydrate triazole tethered 2-pyridyl-benzimidazole ligands: Synthesis of their palladium (II) complexes and antimicrobial activities

Deepthi, S., Ramesh, P., Trivedi, R., Buddana, S. K., & Prakasham, R. S. (2015) · Inorganica Chimica Acta · doi:10.1016/j.ica.2015.06.027 · Cited by 23 · see citing works

Click inspired synthesis of triazole-linked vanillin glycoconjugates

Dwivedi, P., Mishra, K. B., Pritika, Mishra, B. B., & Tiwari, V. K. (2016) · Glycoconjugate Journal · doi:10.1007/s10719-016-9729-4 · Cited by 23 · see citing works

Chapter 1. Privileged Scaffolds in Medicinal Chemistry: An Introduction

Barreiro, E. J. (2015) · RSC drug discovery/RSC drug discovery series · doi:10.1039/9781782622246-00001 · Cited by 22 · see citing works

Novel anticancer agent, SQAP, binds to focal adhesion kinase and modulates its activity

Izaguirre-Carbonell, J., Kawakubo, H., Murata, H., Tanabe, A., Takeuchi, T., Kusayanagi, T., Tsukuda, S., Hirakawa, T., Iwabata, K., Kanai, Y., et al. (2015) · Scientific Reports · doi:10.1038/srep15136 · Cited by 22 · see citing works

Potent and specific sialyltransferase inhibitors: imino-linked 5a′-carbadisaccharides

Okazaki, K., Nishigaki, S., Ishizuka, F., Kajihara, Y., & Ogawa, S. (2003) · Organic & Biomolecular Chemistry · doi:10.1039/b304695h · Cited by 20 · see citing works

Synthesis and molecular modelling studies of novel carbapeptide analogs for inhibition of HIV-1 protease

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Anionic glycolipids related to glucuronosyldiacylglycerol inhibit protein kinase Akt

Vetro, M., Costa, B., Donvito, G., Arrighetti, N., Cipolla, L., Perego, P., Compostella, F., Ronchetti, F., & Colombo, D. (2014) · Organic & Biomolecular Chemistry · doi:10.1039/c4ob01602e · Cited by 18 · see citing works

Cell cycle arrest, apoptosis and autophagy induced by iminosugars on K562 cells

Zhu, J., Zhou, Y., Wang, G., Tai, G., & Ye, X. (2014) · European Journal of Pharmacology · doi:10.1016/j.ejphar.2014.03.013 · Cited by 16 · see citing works

Oral empagliflozin-loaded tri-layer core-sheath fibers fabricated using tri-axial electrospinning: Enhanced in vitro and in vivo antidiabetic performance

Güler, E., Hazar‐Yavuz, A. N., Tatar, E., Haidari, M. M., Ozcan, G. S., Duruksu, G., Graça, M. P. F., Kalaskar, D. M., Gündüz, O., & Çam, M. E. (2023) · International Journal of Pharmaceutics · doi:10.1016/j.ijpharm.2023.122716 · Cited by 41 · see citing works

GANAB and N-Glycans Substrates Are Relevant in Human Physiology, Polycystic Pathology and Multiple Sclerosis: A Review

De Masi, R., & Orlando, S. (2022) · International Journal of Molecular Sciences · doi:10.3390/ijms23137373 · Cited by 20 · see citing works

Rationalizing Graph Neural Networks with Data Augmentation

Liu, G., Inae, E., Luo, T., & Jiang, M. (2023) · ACM Transactions on Knowledge Discovery from Data · doi:10.1145/3638781 · Cited by 15 · see citing works

Stereoselective Synthesis and Immunological Evaluation of Common O‐antigen of P. mirabilis OE and P. vulgaris TG103

Wu, X., Lai, J., Yang, K., Xue, Y., Liao, J., Wang, L., Sun, J., Jing Hua, H. U., Yin, J., & Zhang, Q. (2022) · Chinese Journal of Chemistry · doi:10.1002/cjoc.202200638 · Cited by 11 · see citing works

Recent advances in stereoselective intramolecular O-glycosylation

Jaiswal, M. K., Sharma, A., Tiwari, V. K., & Schmidt, R. R. (2023) · Elsevier eBooks · doi:10.1016/b978-0-323-91729-2.00020-3 · Cited by 8 · see citing works

Electrosynthesis of Sugar Derivatives

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Carbohydrates mimetics: enzyme inhibitors and target molecules in several diseases

Manzano, V. E., Lobo, C. A. C., & Repetto, E. (2021) · Elsevier eBooks · doi:10.1016/b978-0-323-85759-8.00024-5 · Cited by 5 · see citing works

An expeditious one-pot synthesis of thiourea derivatives of carbohydrates from sugar azides

Mishra, K. B., Rajkhowa, S., & Tiwari, V. K. (2020) · Journal of Carbohydrate Chemistry · doi:10.1080/07328303.2020.1822997 · Cited by 5 · see citing works

Glycosylation Modulation Dictates Trafficking and Interaction of SARS-CoV-2 S1 Subunit and ACE2 in Intestinal Epithelial Caco-2 Cells

Khoury, M. E., Wanes, D., Lynch-Miller, M., Hoter, A., & Naim, H. Y. (2024) · Biomolecules · doi:10.3390/biom14050537 · Cited by 4 · see citing works

Copper-Catalyzed Photocatalyst-Free Radical N -Glycosylation

Lai, J., Zhu, Y., Huang, Z., Liu, D., Liu, C., Wang, Z., Wang, L., Chen, F., & Zhang, Q. (2026) · ACS Catalysis · doi:10.1021/acscatal.6c00469 · Cited by 3 · see citing works

Synthesis of Methylene Tetrahydrofurane‐Fused Carbohydrates

Ahmadian-Moghaddam, M., Reintjens, N. R. M., Witte, M. D., & Minnaard, A. J. (2023) · European Journal of Organic Chemistry · doi:10.1002/ejoc.202300281 · Cited by 3 · see citing works

Carbohydrate-based chiral organocatalysts

Tiwari, V. K., & Pellissier, H. (2023) · Elsevier eBooks · doi:10.1016/b978-0-323-91729-2.00021-5 · Cited by 3 · see citing works

Synthesis of 1,2,3-Triazole and Tetrazole Appended Glycoconjugates Based on 3,6-Anhydroglucofuranose via Click Reaction

Das, S. K., Hore, R., Paria, S., Dcosta, G., Kundu, M., & Maity, J. (2025) · ACS Omega · doi:10.1021/acsomega.5c02564 · Cited by 2 · see citing works

N-Alkyl Derivatives of Deoxynojirimycin (DNJ) as Antiviral Agents: Overview and Update

Checconi, P., Iacopetta, D., Catalano, A. A., Ceramella, J., Cavalluzzi, M. M., Mariconda, A., Marsico, S., Aquaro, S., Longo, P., Sinicropi, M. S., et al. (2026) · Molecules · doi:10.3390/molecules31030399 · Cited by 2 · see citing works

Synthesis of methyl 3,4-anhydro-6-bromo-2-O-tert-butyldimethylsilyl-6-deoxy-α-d-allopyranoside from α-d-glucose

Glisin, D., Jovanovic, O., Stojanović, G., Zivkovic, A., Stojanovic, D., Pavlovic, M., & ARSIC, B. B. (2024) · Journal of the Serbian Chemical Society · doi:10.2298/jsc230831049g · Cited by 1 · see citing works

Synthesis, fabrication and characterization of composite scaffolds employing sodium alginate, nanoclay and hydroxyapatite for articular cartilage tissue engineering

Shahbazi, P., Abdouss, M., Naeimi, M., Darbemamieh, G., & Jafari‐Nodoushan, M. (2025) · Carbohydrate Polymer Technologies and Applications · doi:10.1016/j.carpta.2025.100771

Dedicated issue of ‘Carbohydrate Research’ as part of celebration of 90th birth anniversary of Prof. (em.) Dr. Richard R. Schmidt

Tiwari, V. K. (2025) · Carbohydrate Research · doi:10.1016/j.carres.2025.109701

Carbohydrate based Potential Chemotherapeutic Agents: Recent Developments and their Scope in Future Drug Discovery

Tiwari, V. K., Mishra, R. C., Sharma, A., & Tripathi, R. P. (2012) · Mini-Reviews in Medicinal Chemistry · doi:10.2174/138955712803832654 · Cited by 96 · see citing works

Development of Diverse Range of Biologically Relevant Carbohydrate‐Containing Molecules: Twenty Years of Our Journey**

Tiwari, V. K. (2021) · The Chemical Record · doi:10.1002/tcr.202100058 · Cited by 44 · see citing works

Carbohydrate-Based Therapeutics

Mishra, S., Upadhaya, K., Mishra, K. B., Shukla, A. K., Tripathi, R. P., & Tiwari, V. K. (2016) · Studies in natural products chemistry · doi:10.1016/b978-0-444-63601-0.00010-7 · Cited by 47 · see citing works

Carbohydrates as Scaffolds in Drug Discovery

Meutermans, W. D. F., Le, G. T., & Becker, B. (2006) · ChemMedChem · doi:10.1002/cmdc.200600150 · Cited by 122 · see citing works

THE ROLE OF CARBOHYDRATES IN DRUG DISCOVERY: FROM NATURAL SUGARS TO SYNTHETIC GLYCOMIMETICS

Amhanokhai, E. A. (2026) · Zenodo (CERN European Organization for Nuclear Research) · doi:10.5281/zenodo.23397617