Varenicline: An α4β2 Nicotinic Receptor Partial Agonist for Smoking Cessation

Cited by (960)

Items 901–960 of 960

  1. The Pharmacist's Role in Smoking Cessation
    Jeannette Y. Wick · 2008 · The Consultant Pharmacist
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  5. Agents for Treatment of Withdrawal and Dependency: Varenicline
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  6. Function and pharmacology of neuronal nAChRs
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  7. EPIDEMIOLOGIA PALENIA TYTONIU I METODY EFEKTYWNIE WSPIERAJĄCE WALKĘ Z UZALEŻNIENIEM OD NIKOTYNY
    Wojciech Wahl, Dorota Jędrzejczyk-Okońska, Adam Fronczak · 2019 · Prospects in Pharmaceutical Sciences
  8. Eficácia do uso de marcadores genéticos na escolha do tratamento farmacológico do tabagismo com bupropiona e vareniclina e implicações na combinação das drogas: estudo randomizado, controlado
    Patrícia Viviane Gaya · 2023 · Digital Library of Theses and Dissertations (Universidade de São Paulo)
  9. Construction of Bridged Benzazepines via Photo‐Induced Dearomatization
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  10. Modulators of nicotine reward and reinforcement
    Brandon J. Henderson, Samuel Tetteh-Quarshie, Nathan A. Olszewski · 2024 · Advances in pharmacology
  11. Gestion périopératoire des cigarettes conventionnelles et électroniques. Actualisation 2023. Une revue narrative de la littérature
    Margaux Mestdag, Stéphanie Degey, Eric P. DEFLANDRE · 2024 · Revue des Maladies Respiratoires
  12. Retrospective evaluation of COVID-19 incidence during smoking cessation treatment with varenicline
    Elif Barış, Gökçen Ömeroğlu Şi̇mşek, Aylin Arıcı, Mukaddes Gümüştekin, Oğuz Kılınç, Metiner Tosun · 2024 · Celal Bayar Üniversitesi Sağlık Bilimleri Enstitüsü Dergisi
  13. Chapter 54. Treatment of Substance Use Disorders
    Brian J. Sherman, Karen J. Hartwell, Aimee L. McRae‐Clark, Alexandra Herron, Kathleen T. Brady · 2024 · American Psychiatric Association Publishing eBooks
  14. Roles of metabotropic signaling of nicotine receptors in the development and maintenance of nicotine reward through regulation of dopamine D 3 receptor expression
    Dooti Kundu, Srijan Acharya, Shujie Wang, Yongkai Cao, Hee Jin Kim, Jae Hoon Cheong, Kyeong‐Man Kim · 2024 · Journal of Neurochemistry
  15. Allosteric Control of Super-Agonism in a Ligand-Gated Ion Channel
    Franco Viscarra, Teresa Minguez, Isabel Bermúdez, Philip Charles Biggin · 2025 · bioRxiv (Cold Spring Harbor Laboratory)
  16. Deciphering the Activation Mechanism and Internal Signaling Pathways of Dopamine Receptor D1 bound with Various Ligands via Molecular Simulations
    Xing-Yan Lai, Hao‐Jen Hsu, Chun‐Chun Chang · 2025 · Annual International Conference of the IEEE Engineering in Medicine and Biology Society (EMBC)
  17. Chapter 6.2 Use of microdialysis in drug discovery and development: industry and regulatory perspectives
    Hans Rollema, Chandra S. Chaurasia · 2006 · Handbook of behavioral neuroscience
  18. A Pharmacological Update and Safety Analysis of Medications for Smoking Cessation: Which Ones to Use?
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  19. Understanding Nicotine Addiction: Personalizing Therapy for Smoking Cessation
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  20. Cytisine—New Challenges of a Well-Known Drug in the Treatment of Nicotine Addiction
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  21. Time-varying mediated effects of the nicotine patch on smoking before and after a quit attempt when it is added to varenicline and counseling
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  25. Functionalization of fused N ‐heterocyclic frameworks using organometallic reagents: Reactivity, selectivity, and biological application
    Jenu Navyatha, Selvam Vasanth, Palanisamy Sowntharya, Pitchamuthu Amaladass, Vasudevan Dhayalan · 2026 · Bulletin of the Korean Chemical Society
  26. Therapeutic potential of varenicline in neuropsychiatric disorders: insights into its molecular mechanisms
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  27. BindingDB Entry 50039254: A novel series of [3.2.1] azabicyclic biaryl ethers as alpha3beta4 and alpha6/4beta4 nicotinic receptor agonists.
    BindingDB · 2013 · UC San Diego
  28. BindingDB Entry 50044857: Enantiopure Cyclopropane-Bearing Pyridyldiazabicyclo[3.3.0]octanes as Selectivea4ß2-nAChR Ligands.
    BindingDB · 2016 · UC San Diego
  29. BindingDB Entry 50009582: New Rigid Nicotine Analogues, Carrying a Norbornane Moiety, Are Potent Agonists of α7 and α3* Nicotinic Receptors.
    BindingDB · 2021 · UC San Diego
  30. BindingDB Entry 50034073: Docking studies of benzylidene anabaseine interactions witha7 nicotinic acetylcholine receptor (nAChR) and acetylcholine binding proteins (AChBPs): application to the design of relateda7 selective ligands.
    BindingDB · 2012 · UC San Diego
  31. BindingDB Entry 50022743: Seven-membered N-heterocycles as approved drugs and promising leads in medicinal chemistry as well as the metal-free domino access to their scaffolds.
    BindingDB · 2026 · UC San Diego
  32. BindingDB Entry 50042577: Chemistry and pharmacological studies of 3-alkoxy-2,5-disubstituted-pyridinyl compounds as novel selectivea4ß2 nicotinic acetylcholine receptor ligands that reduce alcohol intake in rats.
    BindingDB · 2013 · UC San Diego
  33. BindingDB Entry 50044154: Design, synthesis, and biological evaluation of Erythrina alkaloid analogues as neuronal nicotinic acetylcholine receptor antagonists.
    BindingDB · 2015 · UC San Diego
  34. BindingDB Entry 50048256: Synthesis and biological evaluation of novel hybrids of highly potent and selectivea4ß2-Nicotinic acetylcholine receptor (nAChR) partial agonists.
    BindingDB · 2018 · UC San Diego
  35. BindingDB Entry 50038345: Deconstructing cytisine: The syntheses of (+/-)-cyfusine and (+/-)-cyclopropylcyfusine, fused ring analogs of cytisine.
    BindingDB · 2012 · UC San Diego
  36. BindingDB Entry 50040506: Synthesis and nicotinic acetylcholine receptor in vitro and in vivo pharmacological properties of 2'-fluoro-3'-(substituted phenyl)deschloroepibatidine analogues of 2'-fluoro-3'-(4-nitrophenyl)deschloroepibatidine.
    BindingDB · 2013 · UC San Diego
  37. BindingDB Entry 50028853: Synthesis, binding, and modeling studies of new cytisine derivatives, as ligands for neuronal nicotinic acetylcholine receptor subtypes.
    BindingDB · 2010 · UC San Diego
  38. BindingDB Entry 5532: 7-Azaindole derivatives as potential partial nicotinic agonists.
    BindingDB · 2012 · UC San Diego
  39. BindingDB Entry 50043624: The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor (nAChR) ligands. Part 1: the influence of different hydrogen bond acceptor systems on alkyl and (hetero)aryl substituents.
    BindingDB · 2014 · UC San Diego
  40. BindingDB Entry 50043748: Synthesis and activity of substituted heteroaromatics as positive allosteric modulators fora4ß2a5 nicotinic acetylcholine receptors.
    BindingDB · 2014 · UC San Diego
  41. BindingDB Entry 50037393: In pursuit of alpha4beta2 nicotinic receptor partial agonists for smoking cessation: carbon analogs of (-)-cytisine.
    BindingDB · 2012 · UC San Diego
  42. BindingDB Entry 50041968: Structure-based design, synthesis and structure-activity relationships of dibenzosuberyl- and benzoate-substituted tropines as ligands for acetylcholine-binding protein.
    BindingDB · 2013 · UC San Diego
  43. BindingDB Entry 50040471: Identification of novela4ß2-nicotinic acetylcholine receptor (nAChR) agonists based on an isoxazole ether scaffold that demonstrate antidepressant-like activity.
    BindingDB · 2013 · UC San Diego
  44. BindingDB Entry 50037598: 3,5-Bicyclic aryl piperidines: a novel class of alpha4beta2 neuronal nicotinic receptor partial agonists for smoking cessation.
    BindingDB · 2012 · UC San Diego
  45. BindingDB Entry 50031251: Discovery of 4-(5-methyloxazolo[4,5-b]pyridin-2-yl)-1,4-diazabicyclo[3.2.2]nonane (CP-810,123), a novel alpha 7 nicotinic acetylcholine receptor agonist for the treatment of cognitive disorders in schizophrenia: synthesis, SAR development, and in vivo efficacy in cognition models.
    BindingDB · 2010 · UC San Diego
  46. BindingDB Entry 50004601: Structure-activity studies of diazabicyclo[3.3.0]octane-substituted pyrazines and pyridines as potent α4β2 nicotinic acetylcholine receptor ligands.
    BindingDB · 2020 · UC San Diego
  47. BindingDB Entry 50028566: Diversity-oriented synthesis of a cytisine-inspired pyridone library leading to the discovery of novel inhibitors of Bcl-2.
    BindingDB · 2010 · UC San Diego
  48. BindingDB Entry 50045100: Recent developments in novel antidepressants targetinga4ß2-nicotinic acetylcholine receptors.
    BindingDB · 2016 · UC San Diego
  49. BindingDB Entry 50043453: QM-polarized ligand docking accurately predicts the trend in binding affinity of a series of arylmethylene quinuclidine-like derivatives at thea4ß2 anda3ß4 nicotinic acetylcholine receptors (nAChRs).
    BindingDB · 2014 · UC San Diego
  50. BindingDB Entry 50042476: Ion channels as therapeutic targets: a drug discovery perspective.
    BindingDB · 2013 · UC San Diego
  51. BindingDB Entry 50011567: Pyridine alkaloids with activity in the central nervous system.
    BindingDB · 2022 · UC San Diego
  52. BindingDB Entry 50043556: TBA
    BindingDB · 2014 · UC San Diego
  53. BindingDB Entry 50005284: Pharmacological properties and predicted binding mode of arylmethylene quinuclidine-like derivatives at the α3β4 nicotinic acetylcholine receptor (nAChR).
    BindingDB · 2020 · UC San Diego
  54. BindingDB Entry 50043943: Synthesis, nicotinic acetylcholine receptor binding, and antinociceptive properties of 2'-fluoro-3'-(substituted pyridinyl)-7-deschloroepibatidine analogues.
    BindingDB · 2014 · UC San Diego
  55. BindingDB Entry 50007593: An insight into medicinal chemistry of anticancer quinoxalines.
    BindingDB · 2021 · UC San Diego
  56. BindingDB Entry 50014100: Structure activity relationship (SAR) study identifies a quinoxaline urea analog that modulates IKKβ phosphorylation for pancreatic cancer therapy.
    BindingDB · 2022 · UC San Diego
  57. BindingDB Entry 50033481: Evaluation of structurally diverse neuronal nicotinic receptor ligands for selectivity at the alpha6( *) subtype.
    BindingDB · 2011 · UC San Diego
  58. Regulation and Function of Neuronal Nicotinic Acetylcholine Receptors in Lung Cancer: A Dissertation
    Ma. Reina Improgo · 2011 · eScholarship@UMassChan
  59. Regulation of Neuronal Nicotinic Receptor Expression by Novel Ligands and Mechanisms
    G. Patrick Hussmann · 2012 · DigitalGeorgetown (Georgetown University Library)
  60. Estratégias para a cessação do tabagismo : uma revisão das alternativas terapêuticas
    Marlise Lara Fagundes · 2010 · Lume (Universidade Federal do Rio Grande do Sul)