Critical roles of non-histone protein lysine methylation in human tumorigenesis

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Methylation of H3-Lysine 79 Is Mediated by a New Family of HMTases without a SET Domain

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hDOT1L Links Histone Methylation to Leukemogenesis

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p53 is regulated by the lysine demethylase LSD1

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SET Domain-containing Protein, G9a, Is a Novel Lysine-preferring Mammalian Histone Methyltransferase with Hyperactivity and Specific Selectivity to Lysines 9 and 27 of Histone H3

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A selective inhibitor of EZH2 blocks H3K27 methylation and kills mutant lymphoma cells

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SMYD3 encodes a histone methyltransferase involved in the proliferation of cancer cells

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Inhibition of the LSD1 (KDM1A) demethylase reactivates the all-trans-retinoic acid differentiation pathway in acute myeloid leukemia

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A chemical probe selectively inhibits G9a and GLP methyltransferase activity in cells

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Selective Inhibition of EZH2 by EPZ-6438 Leads to Potent Antitumor Activity in EZH2 -Mutant Non-Hodgkin Lymphoma

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The Occurrence of iε-N-Methyl Lysine in Histones

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Modulation of p53 Function by SET8-Mediated Methylation at Lysine 382

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Validation of a Prognostic Model and the Impact of Mutations in Patients With Lower-Risk Myelodysplastic Syndromes

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NUP98–NSD1 links H3K36 methylation to Hox-A gene activation and leukaemogenesis

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MMSET regulates histone H4K20 methylation and 53BP1 accumulation at DNA damage sites

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ɛ-N-Methyl-lysine in Bacterial Flagellar Protein

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Regulation of NF-κB by NSD1/FBXL11-dependent reversible lysine methylation of p65

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Highly effective combination of LSD1 (KDM1A) antagonist and pan-histone deacetylase inhibitor against human AML cells

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EZH2 Generates a Methyl Degron that Is Recognized by the DCAF1/DDB1/CUL4 E3 Ubiquitin Ligase Complex

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Lysine methylation of the NF-κB subunit RelA by SETD6 couples activity of the histone methyltransferase GLP at chromatin to tonic repression of NF-κB signaling

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Human LSD2/KDM1b/AOF1 Regulates Gene Transcription by Modulating Intragenic H3K4me2 Methylation

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Demethylation of RB Regulator MYPT1 by Histone Demethylase LSD1 Promotes Cell Cycle Progression in Cancer Cells

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Novel Histone Demethylase LSD1 Inhibitors Selectively Target Cancer Cells with Pluripotent Stem Cell Properties

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Methylation of the Retinoblastoma Tumor Suppressor by SMYD2

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Histone Lysine Methyltransferase SETD8 Promotes Carcinogenesis by Deregulating PCNA Expression

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RB1 Methylation by SMYD2 Enhances Cell Cycle Progression through an Increase of RB1 Phosphorylation

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JARID1B Is a Luminal Lineage-Driving Oncogene in Breast Cancer

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