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Transformable nanodrugs for overcoming the biological barriers in the tumor environment during drug delivery
Abstract
Transformable nanodrugs with changeable sizes and shapes allow for overcoming multiple biological barriers for enhanced drug delivery. This review aims to present an overview of the most recent development of smart nanodrugs in this emerging field.
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“First, pH followed by enzyme or GSH cascades, in which mild acidification initiates partial downsizing or loosens the corona before a second stimulus exposes cationic or targeting domains [28].”
From Overcoming tumor microenvironment barriers: transformable and bioinspired nanomedicine strategies for deep tumor penetration (2026) · cites this paper as [28]
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Li, H.-J., Du, J.-Z., Liu, J., Du, X.-J., Shen, S., Zhu, Y.-H., Wang, X., Ye, X., Nie, S., & Wang, J. (2016) · ACS Nano · doi:10.1021/acsnano.6b02326 · Cited by 537
Ultrasound-responsive systems as components for smart materials
Athanassiadis, A. G., Ma, Z., Moreno-Gomez, N., Melde, K., Choi, E., Goyal, R., & Fischer, P. (2022) · Chemical Reviews · doi:10.1021/acs.chemrev.1c00622 · Cited by 293
Transformable Helical Self-Assembly for Cancerous Golgi Apparatus Disruption
Li, R. S., Liu, J., Shi, H., Hu, P. P., Wang, Y., Gao, P. F., Wang, J., Jia, M., Li, H., Li, Y. F., et al. (2021) · Nano Letters · doi:10.1021/acs.nanolett.1c03112 · Cited by 59
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Cited by
Sorted by citations
Sheng, J., Yuan, W., Zhang, M., Chen, Z., Qi, Y., Zhao, Y., & Zhang, S. (2026) · Journal of Nanobiotechnology · doi:10.1186/s12951-026-04028-7 · Cited by 35
Metadata
- Authors
- Li, X., Huang, Z., Liao, Z., Liu, A., & Huo, S.
- Venue
- Nanoscale
- Publisher
- Royal Society of Chemistry (RSC)
- Published
- 2023
- Volume
- 15
- Issue
- 19
- Pages
- 8532-8547
- ISSN
- 2040-3364
- 2040-3372
- Cited by
- 13
- References
- 3
- Language
- en
- Update notices
- correction (2025-05-28)
- Funders
- National Natural Science Foundation of China (82001959)
- Natural Science Foundation of Xiamen Municipality (3502Z20227004)
- Fundamental Research Funds for the Central Universities (20720210102)
- Xiamen University
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