International Union of Pharmacology. LXIV. Estrogen Receptors

Cloning of a novel receptor expressed in rat prostate and ovary.

Kuiper, G. G. J. M., Enmark, E., Pelto‐Huikko, M., Nilsson, S., & Gustafsson, J.-Α. (1996) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.93.12.5925 · Cited by 4,792 · see citing works

Comparison of the Ligand Binding Specificity and Transcript Tissue Distribution of Estrogen Receptors α and β

Kuiper, G. G. J. M., Carlsson, B., Grandien, K., Enmark, E., Häggblad, J., Nilsson, S., & Gustafsson, J.-A. (1997) · Endocrinology · doi:10.1210/endo.138.3.4979 · Cited by 4,442 · see citing works

Interaction of Estrogenic Chemicals and Phytoestrogens with Estrogen Receptor β

Kuiper, G. G. J. M., Lemmen, J. G., Carlsson, B., Corton, J. C., Safe, S. H., van der Saag, P. T., van der Burg, B., & Gustafsson, J.-Å. (1998) · Endocrinology · doi:10.1210/endo.139.10.6216 · Cited by 4,203 · see citing works

Molecular basis of agonism and antagonism in the oestrogen receptor

Brzozowski, A. M., Pike, A. C. W., Dauter, Z., Hubbard, R. E., Bonn, T., Engström, O., Öhman, L., Greene, G. L., Gustafsson, J.-Å., & Carlquist, M. (1997) · Nature · doi:10.1038/39645 · Cited by 3,355 · see citing works

The Protective Effects of Estrogen on the Cardiovascular System

Mendelsohn, M. E., & Karas, R. H. (1999) · New England Journal of Medicine · doi:10.1056/nejm199906103402306 · Cited by 3,108 · see citing works

Estrogen Resistance Caused by a Mutation in the Estrogen-Receptor Gene in a Man

Smith, E. P., Boyd, J., Frank, G. R., Takahashi, H., Cohen, R. M., Specker, B., Williams, T. C., Lubahn, D. B., & Korach, K. S. (1994) · New England Journal of Medicine · doi:10.1056/nejm199410203311604 · Cited by 2,471 · see citing works

Human oestrogen receptor cDNA: sequence, expression and homology to v-erb-A

Green, S., Walter, P., Kumar, V., Krust, A., Bornert, J., Argos, P., & Chambon, P. (1986) · Nature · doi:10.1038/320134a0 · Cited by 2,320 · see citing works

Effects of Tamoxifen vs Raloxifene on the Risk of Developing Invasive Breast Cancer and Other Disease Outcomes<SUBTITLE>The NSABP Study of Tamoxifen and Raloxifene (STAR) P-2 Trial</SUBTITLE>

Vogel, V. G. (2006) · JAMA · doi:10.1001/jama.295.23.joc60074 · Cited by 1,652 · see citing works

Sequence and Expression of Human Estrogen Receptor Complementary DNA

Greene, G. L., Gilna, P., Waterfield, M. D., BAKER, A. J., Hort, Y., & Shine, J. (1986) · Science · doi:10.1126/science.3753802 · Cited by 1,311 · see citing works

Molecular Determinants for the Tissue Specificity of SERMs

Shang, Y., & Brown, M. A. (2002) · Science · doi:10.1126/science.1068537 · Cited by 1,149 · see citing works

Cloning, Chromosomal Localization, and Functional Analysis of the Murine Estrogen Receptor β

Tremblay, G. B., Tremblay, A., Copeland, N. G., Gilbert, D. J., Jenkins, N. A., Labrie, F., & Giguère, V. (1997) · Molecular Endocrinology · doi:10.1210/mend.11.3.9902 · Cited by 866 · see citing works

Differential Response of Estrogen Receptor α and Estrogen Receptor β to Partial Estrogen Agonists/Antagonists

Barkhem, T., Carlsson, B., Nilsson, Y., Enmark, E., Gustafsson, J.-Α., & Nilsson, S. V. (1998) · Molecular Pharmacology · doi:10.1124/mol.54.1.105 · Cited by 770 · see citing works

Pyrazole Ligands: Structure−Affinity/Activity Relationships and Estrogen Receptor-α-Selective Agonists

Stauffer, S. R., Coletta, C. J., Tedesco, R., Nishiguchi, G., Carlson, K. E., Sun, J., Katzenellenbogen, B. S., & Katzenellenbogen, J. A. (2000) · Journal of Medicinal Chemistry · doi:10.1021/jm000170m · Cited by 760 · see citing works

Effects of estrogen plus progestin on health-related quality of life

Hays, J., Ockene, J. K., Brunner, R. L., Kotchen, J. M., Manson, J. E., Patterson, R. E., Aragaki, A. K., Shumaker, S. A., Brzyski, R. G., LaCroix, A. Z., et al. (2003) · New England Journal of Medicine · doi:10.1056/nejmoa030311 · Cited by 686 · see citing works

Estrogen Receptor-β Potency-Selective Ligands: Structure−Activity Relationship Studies of Diarylpropionitriles and Their Acetylene and Polar Analogues

Meyers, M. J., Sun, J., Carlson, K. E., Marriner, G. A., Katzenellenbogen, B. S., & Katzenellenbogen, J. A. (2001) · Journal of Medicinal Chemistry · doi:10.1021/jm010254a · Cited by 678 · see citing works

Human estrogen receptor transactivational capacity is determined by both cellular and promoter context and mediated by two functionally distinct intramolecular regions

Tzukerman, M., Esty, A., Santiso‐Mere, D., Danielian, P. S., Parker, M. G., Stein, R. B., Pike, J. W., & McDonnell, D. P. (1994) · Molecular Endocrinology · doi:10.1210/mend.8.1.8152428 · Cited by 671 · see citing works

A systematic review of genetic polymorphisms and breast cancer risk.

Dunning, A., Healey, C. S., Pharoah, P., Teare, M. D., Ponder, B. A. J., & Easton, D. F. (1999) · PubMed · Cited by 539 · see citing works

The Complete Primary Structure of Human Estrogen Receptor β (hERβ) and Its Heterodimerization with ER αin Vivoandin Vitro

Ogawa, S., Inoue, S., Watanabe, T., Hiroi, H., Orimo, A., Hosoi, T., Ouchi, Y., & Muramatsu, M. (1998) · Biochemical and Biophysical Research Communications · doi:10.1006/bbrc.1997.7893 · Cited by 511 · see citing works

Estrogen receptor interaction with co-activators and co-repressors☆

Klinge, C. M. (2000) · Steroids · doi:10.1016/s0039-128x(99)00107-5 · Cited by 489 · see citing works

Molecular cloning and charcterization of rat estrogen receptor cDNA

Koike, S., Sakai, M., & Muramatsu, M. (1987) · Nucleic Acids Research · doi:10.1093/nar/15.6.2499 · Cited by 489 · see citing works

Abnormal Vascular Function and Hypertension in Mice Deficient in Estrogen Receptor β

Zhu, Y., Bian, Z., Lu, P., Karas, R. H., Bao, L., Cox, D. H., Hodgin, J. B., Shaul, P. W., Thorén, P., Smithies, O., et al. (2002) · Science · doi:10.1126/science.1065250 · Cited by 482 · see citing works

The estrogen receptor: a model for molecular medicine.

Jensen, E. V., & Jordan, V. C. (2003) · PubMed · Cited by 470 · see citing works

Molecular cloning and characterization of human estrogen receptor betacx: a potential inhibitor ofestrogen action in human

Ogawa, S. (1998) · Nucleic Acids Research · doi:10.1093/nar/26.15.3505 · Cited by 448 · see citing works

Identification of a new isoform of the human estrogen receptor‐alpha (hER‐α) that is encoded by distinct transcripts and that is able to repress hER‐α activation function 1

Flouriot, G., Brand, H., Denger, S., Métivier, R., Koš, M., Reid, G., Sonntag‐Buck, V., & Gannon, F. (2000) · The EMBO Journal · doi:10.1093/emboj/19.17.4688 · Cited by 419 · see citing works

Transcriptional activation of genes by 17β-estradiol through estrogen receptor-Sp1 interactions

Safe, S. H. (2001) · Vitamins and hormones · doi:10.1016/s0083-6729(01)62006-5 · Cited by 418 · see citing works

ERβ Inhibits Proliferation and Invasion of Breast Cancer Cells

Lazennec, G., Bresson, D., Lucas, A., Chauveau, C., & Vignon, F. (2001) · Endocrinology · doi:10.1210/endo.142.9.8395 · Cited by 379 · see citing works

Estrogen-Receptor Polymorphisms and Effects of Estrogen Replacement on High-Density Lipoprotein Cholesterol in Women with Coronary Disease

Herrington, D. M., Howard, T. D., Hawkins, G. A., Reboussin, D. M., Xu, J., Zheng, S. L., Brosnihan, K. B., Meyers, D. A., & Bleecker, E. R. (2002) · New England Journal of Medicine · doi:10.1056/nejmoa012952 · Cited by 372 · see citing works

Estrogen Receptor-α Mediates the Protective Effects of Estrogen Against Vascular Injury

Pare, G. J., Krust, A., Karas, R. H., Dupont, S., Aronovitz, M. A., Chambon, P., & Mendelsohn, M. E. (2002) · Circulation Research · doi:10.1161/01.res.0000021114.92282.fa · Cited by 369 · see citing works

Direct Acetylation of the Estrogen Receptor α Hinge Region by p300 Regulates Transactivation and Hormone Sensitivity

Wang, C., Fu, M., Angeletti, R. H., Siconolfi-Baez, L., Reutens, A. T., Albanese, C., Lisanti, M. P., Katzenellenbogen, B. S., Kato, S., Hopp, T., et al. (2001) · Journal of Biological Chemistry · doi:10.1074/jbc.m100800200 · Cited by 365 · see citing works

Structural Organization and Expression of the Mouse Estrogen Receptor

White, R., Lees, J. A., Needham, M., Ham, J., & Parker, M. G. (1987) · Molecular Endocrinology · doi:10.1210/mend-1-10-735 · Cited by 362 · see citing works

Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism

Shiau, A. K., Barstad, D., Radek, J. T., Meyers, M. J., Nettles, K. W., Katzenellenbogen, B. S., Katzenellenbogen, J. A., Agard, D. A., & Greene, G. L. (2002) · Nature Structural Biology · doi:10.1038/nsb787 · Cited by 357 · see citing works

Deletion of estrogen receptors reveals a regulatory role for estrogen receptors-β in bone remodeling in females but not in males

Sims, N. A., Dupont, S., Krust, A., Clément-Lacroix, P., Minet, D., Resche-Rigon, M., Gaillard-Kelly, M., & Baron, R. (2002) · Bone · doi:10.1016/s8756-3282(01)00643-3 · Cited by 354 · see citing works

Cloning, Chromosomal Localization, and Functional Analysis of the Murine Estrogen Receptor

Tremblay, G. B. (1997) · Molecular Endocrinology · doi:10.1210/me.11.3.353 · Cited by 339 · see citing works

Effects of Tamoxifen vs Raloxifene on the Risk of Developing Invasive Breast Cancer and Other Disease Outcomes. The NSABP Study of Tamoxifen and Raloxifene (STAR) P-2 Trial

Vogel, V. G., Costantino, J. P., Wickerham, D. L., Cronin, W. M., Cecchini, R. S., Atkins, J. N., Bevers, T. B., Fehrenbacher, L., Pajon, E. R., Wade, J. L., et al. (2006) · Obstetrical & Gynecological Survey · doi:10.1097/01.ogx.0000238648.23538.42 · Cited by 329 · see citing works

Effects of anti-estrogens on bone in castrated and intact female rats

Jordan, V. C., Phelps, E., & Lindgren, J. (1987) · Breast Cancer Research and Treatment · doi:10.1007/bf01806132 · Cited by 323 · see citing works

Novel Ligands that Function as Selective Estrogens or Antiestrogens for Estrogen Receptor-α or Estrogen Receptor-β*

Sun, J., Meyers, M. J., Fink, B. E., Rajendran, R. R., Katzenellenbogen, J. A., & Katzenellenbogen, B. S. (1999) · Endocrinology · doi:10.1210/endo.140.2.6480 · Cited by 315 · see citing works

Coregulators in Nuclear Estrogen Receptor Action: From Concept to Therapeutic Targeting

Hall, J. M. (2005) · Molecular Interventions · doi:10.1124/mi.5.6.7 · Cited by 291 · see citing works

Selective estrogen receptor modulators (SERMs): Mechanisms of anticarcinogenesis and drug resistance

Lewis, J. S., & Jordan, V. C. (2005) · Mutation research. Fundamental and molecular mechanisms of mutagenesis · doi:10.1016/j.mrfmmm.2005.02.028 · Cited by 282 · see citing works

Immune Modulation in Multiple Sclerosis Patients Treated with the Pregnancy Hormone Estriol

Soldan, S. S., Retuerto, A. I. A., Sicotte, N. L., & Voskuhl, R. R. (2003) · The Journal of Immunology · doi:10.4049/jimmunol.171.11.6267 · Cited by 277 · see citing works

Minireview: Genomic Organization of the Human ERα Gene Promoter Region

Koš, M., Reid, G., Denger, S., & Gannon, F. (2001) · Molecular Endocrinology · doi:10.1210/mend.15.12.0731 · Cited by 267 · see citing works

A hypersensitive estrogen receptor-alpha mutation in premalignant breast lesions.

Fuqua, S. A. W., Wiltschke, C., ZHANG, Q. X., Borg, Å., Castles, C. G., Friedrichs, W. E., Hopp, T., Hilsenbeck, S. G., Mohsin, S. K., O'Connell, P., et al. (2000) · PubMed · Cited by 234 · see citing works

Update on estrogen signaling

Weihua, Z., Andersson, S., Cheng, G., Simpson, E. R., Warner, M. N., & Gustafsson, J.-Α. (2003) · FEBS Letters · doi:10.1016/s0014-5793(03)00436-8 · Cited by 220 · see citing works

Estrogen receptor β regulates epithelial cellular differentiation in the mouse ventral prostate

Imamov, O., Morani, A., Shim, G.-J., Omoto, Y., Thulin-Andersson, C., Warner, M. N., & Gustafsson, J.-Α. (2004) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.0403041101 · Cited by 208 · see citing works

Estrogen Receptor-α Knockout Mice Exhibit Resistance to the Developmental Effects of Neonatal Diethylstilbestrol Exposure on the Female Reproductive Tract

Couse, J. F., Dixon, D., Yates, M. M., Moore, A. B., Ma, L., Maas, R. L., & Korach, K. S. (2001) · Developmental Biology · doi:10.1006/dbio.2001.0413 · Cited by 192 · see citing works

Role of ovarian hormones in the long-term control of glucose homeostasis

Bailey, C. J., & Ahmed-Sorour, H. (1980) · Diabetologia · doi:10.1007/bf00281829 · Cited by 186 · see citing works

Expression of wild-type estrogen receptor beta and variant isoforms in human breast cancer.

Fuqua, S. A. W., Schiff, R., Parra, I., Friedrichs, W. E., Su, J. L., McKee, D. D., Slentz‐Kesler, K., Moore, L. B., Willson, T. M., & Moore, J. T. (1999) · PubMed · Cited by 177 · see citing works

ER Inhibits Proliferation and Invasion of Breast Cancer Cells

Lazennec, G. (2001) · Endocrinology · doi:10.1210/en.142.9.4120 · Cited by 170 · see citing works

Expression of estrogen receptor β isoforms in normal breast epithelial cells and breast cancer: regulation by methylation

Zhao, C., Lam, E. W. ‐., Sunters, A., Enmark, E., Bella, M. T. D., Coombes, R. C., Gustafsson, J.-Α., & Dahlman‐Wright, K. (2003) · Oncogene · doi:10.1038/sj.onc.1207100 · Cited by 168 · see citing works

Association of Estrogen Receptor β Gene Polymorphism with Bone Mineral Density

Ogawa, S., Hosoi, T., Shiraki, M., Orimo, H., Emi, M., Muramatsu, M., Ouchi, Y., & Inoue, S. (2000) · Biochemical and Biophysical Research Communications · doi:10.1006/bbrc.2000.2285 · Cited by 161 · see citing works

Identification of a splice variant of the rat estrogen receptor β gene

Chu, S., & Fuller, P. J. (1997) · Molecular and Cellular Endocrinology · doi:10.1016/s0303-7207(97)00133-0 · Cited by 157 · see citing works

Functional Differences between the Amino-Terminal Domains of Estrogen Receptors α and β

Delaunay, F., Pettersson, K., Tujague, M., & Gustafsson, J.-Å. (2000) · Molecular Pharmacology · doi:10.1124/mol.58.3.584 · Cited by 155 · see citing works

Phosphorylation of Estrogen Receptor α Blocks Its Acetylation and Regulates Estrogen Sensitivity

Cui, Y., Zhang, M., Pestell, R. G., Curran, E. M., Welshons, W. V., & Fuqua, S. A. W. (2004) · Cancer Research · doi:10.1158/0008-5472.can-04-2126 · Cited by 154 · see citing works

Systematic Mutation Screening of the Estrogen Receptor Beta Gene in Probands of Different Weight Extremes: Identification of Several Genetic Variants

Rosenkranz, K., Hinney, A., Ziegler, A., Hermann, H., Fichter, M., Mayer, H. G., Siegfried, W., Young, J., Remschmidt, H., & Hebebrand, J. (1998) · The Journal of Clinical Endocrinology & Metabolism · doi:10.1210/jcem.83.12.5471 · Cited by 147 · see citing works

Estrogen Receptor α Mediates Estrogen’s Immune Protection in Autoimmune Disease

Liu, H.-B., Loo, K. K., Palaszynski, K. M., Ashouri, J. F., Lubahn, D. B., & Voskuhl, R. R. (2003) · The Journal of Immunology · doi:10.4049/jimmunol.171.12.6936 · Cited by 144 · see citing works

Differential regulation of the human progesterone receptor gene through an estrogen response element half site and Sp1 sites

Petz, L. N., Ziegler, Y., Schultz, J. R., Kim, H., Kemper, J. K., & Nardulli, A. M. (2004) · The Journal of Steroid Biochemistry and Molecular Biology · doi:10.1016/j.jsbmb.2003.11.008 · Cited by 142 · see citing works

DNA hypermethylation: when tumour suppressor genes go silent

Garinis, G. A., Patrinos, G., Spanakis, N. E., & Menounos, P. (2002) · Human Genetics · doi:10.1007/s00439-002-0783-6 · Cited by 138 · see citing works

Estrogen Receptor Subtype-Selective Ligands: Asymmetric Synthesis and Biological Evaluation of cis- and trans-5,11-Dialkyl- 5,6,11,12-tetrahydrochrysenes

Meyers, M. J., Sun, J., Carlson, K. E., Katzenellenbogen, B. S., & Katzenellenbogen, J. A. (1999) · Journal of Medicinal Chemistry · doi:10.1021/jm990101b · Cited by 137 · see citing works

Identification of pathway-selective estrogen receptor ligands that inhibit NF-κB transcriptional activity

Chadwick, C. C., Chippari, S. M., Matelan, E. M., Borges-Marcucci, L., Eckert, A. M., Keith, J. C., Albert, L. M., Leathurby, Y., Harris, H. A., Bhat, R. A., et al. (2005) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.0405841102 · Cited by 137 · see citing works

A Novel Isoform of Rat Estrogen Receptor Beta with 18 Amino Acid Insertion in the Ligand Binding Domain as a Putative Dominant Negative Regulator of Estrogen Action

Maruyama, K., Endoh, H., Sasaki-Iwaoka, H., Kanou, H., Shimaya, E., Hashimoto, S., Kato, S., & Kawashima, H. (1998) · Biochemical and Biophysical Research Communications · doi:10.1006/bbrc.1998.8590 · Cited by 136 · see citing works

Recent Use of Oral Contraceptives and the Risk of Multiple Sclerosis

Alonso, Á., Jick, S. S., Olek, M. J., Ascherio, A., Jick, H., & Hernán, M. Á. (2005) · Archives of Neurology · doi:10.1001/archneur.62.9.1362 · Cited by 136 · see citing works

Characterization of the Physical Interaction between Estrogen Receptor α and JUN Proteins

Teyssier, C., Belguise, K., Galtier, F., & Chalbos, D. (2001) · Journal of Biological Chemistry · doi:10.1074/jbc.m101806200 · Cited by 130 · see citing works

Estrogens and menopause: pharmacology of conjugated equine estrogens and their potential role in the prevention of neurodegenerative diseases such as Alzheimer’s

Bhavnani, B. R. (2003) · The Journal of Steroid Biochemistry and Molecular Biology · doi:10.1016/s0960-0760(03)00220-6 · Cited by 129 · see citing works

The menopause and obesity

Lovejoy, J. C. (2003) · Primary Care: Clinics in Office Practice · doi:10.1016/s0095-4543(03)00012-5 · Cited by 128 · see citing works

Estrogen Receptor Knockout Mice as a Model for Endocrine Research

Walker, V. R., & Korach, K. S. (2004) · ILAR Journal · doi:10.1093/ilar.45.4.455 · Cited by 128 · see citing works

Quantitative analysis of estrogen receptor-? mRNA and its variants in human breast cancers

Iwao, K., Miyoshi, Y., Egawa, C., Ikeda, N., & Noguchi, S. (2000) · International Journal of Cancer · doi:10.1002/1097-0215(20001201)88:5 · Cited by 124 · see citing works

Association of the Estrogen Receptor α Gene Polymorphisms with Sporadic Alzheimer's Disease

Brandi, M. L., Becherini, L., Gennari, L., Racchi, M., Bianchetti, A., Nacmias, B., Sorbi, S., Mecocci, P., Senin, U., & Govoni, S. M. (1999) · Biochemical and Biophysical Research Communications · doi:10.1006/bbrc.1999.1665 · Cited by 121 · see citing works

Estrogen receptor-α mediates the detrimental effects of neonatal diethylstilbestrol (DES) exposure in the murine reproductive tract

Couse, J. F., & Korach, K. S. (2004) · Toxicology · doi:10.1016/j.tox.2004.06.046 · Cited by 119 · see citing works

Impact of Estrogen Therapy on Alzheimer??s Disease

Brinton, R. D. (2004) · CNS Drugs · doi:10.2165/00023210-200418070-00001 · Cited by 106 · see citing works

Cloning and Characterization of Human Estrogen Receptor β Promoter

Li, L., Yeh, C., Nojima, D., & Dahiya, R. (2000) · Biochemical and Biophysical Research Communications · doi:10.1006/bbrc.2000.3363 · Cited by 104 · see citing works

Toremifene and tamoxifen are equally effective for early-stage breast cancer: first results of International Breast Cancer Study Group Trials 12-93 and 14-93

1 (2004) · Annals of Oncology · doi:10.1093/annonc/mdh463 · Cited by 101 · see citing works

Is the Estrogen Controversy Over? Deconstructing the Women's Health Initiative Study: A Critical Evaluation of the Evidence

Harman, S. M., Naftolin, F. N., Brinton, E. A., & Judelson, D. R. (2005) · Annals of the New York Academy of Sciences · doi:10.1196/annals.1347.004 · Cited by 95 · see citing works

Novel Ligands that Function as Selective Estrogens or Antiestrogens for Estrogen Receptor- or Estrogen Receptor-

Sun, J. (1999) · Endocrinology · doi:10.1210/en.140.2.800 · Cited by 92 · see citing works

Association of estrogen receptor β (ESR2) gene polymorphism with blood pressure

Ogawa, S., Emi, M., Shiraki, M., Hosoi, T., Ouchi, Y., & Inoue, S. (2000) · Journal of Human Genetics · doi:10.1007/s100380070002 · Cited by 87 · see citing works

17 -Estradiol Antiinflammatory Activity in Carrageenan-Induced Pleurisy

Cuzzocrea, S., Santagati, S., Sautebin, L., Mazzon, E., Calabrò, G., Serraino, I., Caputi, A. P., & Maggi, A. C. (2000) · Endocrinology · doi:10.1210/endo.141.4.7404 · Cited by 85 · see citing works

Interaction and Dissociation by Ligands of Estrogen Receptor and Hsp90: The Antiestrogen RU 58668 Induces a Protein Synthesis-Dependent Clustering of the Receptor in the Cytoplasm

Leclerc, J., Meng, X., Delahaye, F., Leclerc, P., Baulieu, É.-É., & CATELLI, M. G. (1998) · Molecular Endocrinology · doi:10.1210/mend.12.6.0121 · Cited by 78 · see citing works

Baseline characteristics of participants in the Raloxifene Use for The Heart (RUTH) trial

WENGER, N. K., Barrett-Connor, E. L., Collins, P. D., Grady, D. G., Kornitzer, M., Mosca, L. J., Sashegyi, A. I., Baygani, S., Anderson, P. W., & Moscarelli, E. (2002) · The American Journal of Cardiology · doi:10.1016/s0002-9149(02)02835-7 · Cited by 76 · see citing works

Association of estrogen receptor β gene polymorphisms with bulimic disease in women

Nilsson, M., Naessén, S., Dahlman, I. A., Hirschberg, A. L., Gustafsson, J., & Dahlman‐Wright, K. (2003) · Molecular Psychiatry · doi:10.1038/sj.mp.4001402 · Cited by 75 · see citing works

Minireview: Genomic Organization of the Human ER Gene Promoter Region

Koš, M. (2001) · Molecular Endocrinology · doi:10.1210/me.15.12.2057 · Cited by 75 · see citing works

Human estrogen receptor messenger RNA variants in both normal and tumor breast tissues

Gotteland, M., Desauty, G., Delarue, J. C., Liu, L., & May, E. (1995) · Molecular and Cellular Endocrinology · doi:10.1016/0303-7207(95)03576-s · Cited by 72 · see citing works

Expression of alternatively spliced estrogen receptor alpha mRNAs is increased in breast cancer tissues

Poola, I., & Speirs, V. (2001) · The Journal of Steroid Biochemistry and Molecular Biology · doi:10.1016/s0960-0760(01)00118-2 · Cited by 65 · see citing works

Dinucleotide repeat polymorphism in the human estrogen receptor (ESR) gene

SENNO, L. D., Aguiari, G., & Piva, R. (1992) · Human Molecular Genetics · doi:10.1093/hmg/1.5.354 · Cited by 60 · see citing works

Role of Ovarian Hormones in the Long-Term Control of Glucose Homeostasis

Ahmed-Sorour, H., & Bailey, C. J. (2008) · Hormone Research · doi:10.1159/000179307 · Cited by 60 · see citing works

The estrogen receptor-α A908G (K303R) mutation occurs at a low frequency in invasive breast tumors: results from a population-based study

Conway, K., Parrish, E., Edmiston, S. N., Tolbert, D., Tse, C., Geradts, J., Livasy, C., Singh, H. K., Newman, B. M., & Millikan, R. C. (2005) · Breast Cancer Research · doi:10.1186/bcr1315 · Cited by 57 · see citing works

Identification of a Functional Imperfect Estrogen-Responsive Element in the 5‘-Promoter Region of the Human Cathepsin D Gene

Wang, F., Porter, W. W., Xing, W., Archer, T., & Safe, S. H. (1997) · Biochemistry · doi:10.1021/bi963100j · Cited by 55 · see citing works

Differential activation of wild-type and variant forms of estrogen receptor α by synthetic and natural estrogenic compounds using a promoter containing three estrogen-responsive elements

Yoon, K., Pallaroni, L., Stoner, M. A., Gaido, K. W., & Safe, S. H. (2001) · The Journal of Steroid Biochemistry and Molecular Biology · doi:10.1016/s0960-0760(01)00070-x · Cited by 53 · see citing works

Estrogen Receptor β: Mine Is Longer Than Yours?a

Leygue, E., Dotzlaw, H., Lü, B., Glor, C., Watson, P. H., & Murphy, L. C. (1998) · The Journal of Clinical Endocrinology & Metabolism · doi:10.1210/jcem.83.10.5187-1 · Cited by 50 · see citing works

pS2Gene Expression in HepG2 cells: Complex Regulation through Crosstalk between the Estrogen Receptor α, an Estrogen-Responsive Element, and the Activator Protein 1 Response Element

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