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Transforming growth factor‐α mediates estrogen‐induced upregulation of glutamate transporter GLT‐1 in rat primary astrocytes

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The nuclear localization signal is required for nuclear GPER translocation and function in breast Cancer-Associated Fibroblasts (CAFs)

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Integrated Bioinformatics, Environmental Epidemiologic and Genomic Approaches to Identify Environmental and Molecular Links between Endometriosis and Breast Cancer

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The Neurosteroid Progesterone Underlies Estrogen Positive Feedback of the LH Surge

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Minireview: Steroidogenic Factor 1: Its Roles in Differentiation, Development, and Disease

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The G protein-coupled estrogen receptor as a modulator of neoplastic transformation

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G protein-coupled estrogen receptor 1 (GPER, GPR 30) in normal human endometrium and early pregnancy decidua

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G Protein-Coupled Estrogen Receptor Mediates Cell Proliferation through the cAMP/PKA/CREB Pathway in Murine Bone Marrow Mesenchymal Stem Cells

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Activation of GPR30 inhibits cardiac fibroblast proliferation

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Low-dose Bisphenol-A regulates inflammatory cytokines through GPR30 in mammary adipose cells

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The effect of tamoxifen and raloxifene on estrogen metabolism and endometrial cancer risk

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Structure of Liver Receptor Homolog-1 (NR5A2) with PIP3 hormone bound in the ligand binding pocket

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Possible role of phytoestrogens in breast cancer via GPER-1/GPR30 signaling

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Roles of estrogen receptors alpha and beta in sexually dimorphic neuroprotection against glutamate toxicity

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Selective GPER activation decreases proliferation and activates apoptosis in tumor Leydig cells

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LRH-1 Governs Vital Transcriptional Programs in Endocrine-Sensitive and -Resistant Breast Cancer Cells

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G Protein-Coupled Estrogen Receptor in Energy Homeostasis and Obesity Pathogenesis

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Racial disparities in histopathologic characteristics of uterine cancer are present in older, not younger blacks in an equal-access environment

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Antiproliferation Activity of a Small Molecule Repressor of Liver Receptor Homolog 1

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Icariin modulates mitochondrial function and apoptosis in high glucose-induced glomerular podocytes through G protein-coupled estrogen receptors

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Molecular Characterization of Membrane Steroid Receptors in Hormone-Sensitive Cancers

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The G Protein-Coupled Receptor GPR30 Mediates the Nontranscriptional Effect of Estrogen on the Activation of PI3K/Akt Pathway in Endometrial Cancer Cells

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The G protein-coupled estrogen receptor 1 (GPER/GPR30) does not predict survival in patients with ovarian cancer

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Regulation of ERRα Gene Expression by Estrogen Receptor Agonists and Antagonists in SKBR3 Breast Cancer Cells: Differential Molecular Mechanisms Mediated by G Protein-Coupled Receptor GPR30/GPER-1

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IQGAP1 is a phosphoinositide effector and kinase scaffold

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A common hypofunctional genetic variant of GPER is associated with increased blood pressure in women

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Tamoxifen activates Nrf2-dependent SQSTM1 transcription to promote endometrial hyperplasia

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Expression of the G protein-coupled estrogen receptor (GPER) in endometriosis: a tissue microarray study

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G protein-coupled estrogen receptor (GPER) mediates NSCLC progression induced by 17β-estradiol (E2) and selective agonist G1

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Repression of mammary adipogenesis by genistein limits mammosphere formation of human MCF-7 cells

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Role of GPR30 in endometrial pathology after tamoxifen for breast cancer

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Activation of G protein-coupled receptor 30 by thiodiphenol promotes proliferation of estrogen receptor α-positive breast cancer cells

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Pathological functions of hypoxia in endometriosis

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Vascular effects of aldosterone: Sorting out the receptors and the ligands

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Estrogen Enhances Linkage in the Vascular Endothelial Calmodulin Network via a Feedforward Mechanism at the G Protein-coupled Estrogen Receptor 1

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Pharmacological, Mechanistic, and Pharmacokinetic Assessment of Novel Melatonin-Tamoxifen Drug Conjugates as Breast Cancer Drugs

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Unraveling the mechanisms underlying the rapid vascular effects of steroids: sorting out the receptors and the pathways

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STX, a Novel Nonsteroidal Estrogenic Compound, Induces Rapid Action in Primate GnRH Neuronal Calcium Dynamics and Peptide Release

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Neuroprotective action of acute estrogens: Animal models of brain ischemia and clinical implications

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Estrogens Induce Rapid Cytoskeleton Re-Organization in Human Dermal Fibroblasts via the Non-Classical Receptor GPR30

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Aldosterone mediates metastatic spread of renal cancer via the G protein‐coupled estrogen receptor (GPER)

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Diacylglycerol kinase α mediates 17-β-estradiol-induced proliferation, motility, and anchorage-independent growth of Hec-1A endometrial cancer cell line through the G protein-coupled estrogen receptor GPR30

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Phospholipid regulation of the nuclear receptor superfamily

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4-Hydroxytamoxifen-stimulated processing of cyclin E is mediated via G protein-coupled receptor 30 (GPR30) and accompanied by enhanced migration in MCF-7 breast cancer cells

Li, Y., Chen, Y., Zhu-xia, Z., Liu, X., Yang, L., Wan, L., Lei, T., & Wang, X. (2013) · Toxicology · doi:10.1016/j.tox.2013.04.012 · Cited by 36 · see citing works

G-protein-coupled receptor 30-mediated antiapoptotic effect of estrogen on spinal motor neurons following injury and its underlying mechanisms

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Inhibition of GPR30 by estriol prevents growth stimulation of triple-negative breast cancer cells by 17β-estradiol

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Understanding the molecular basis of agonist/antagonist mechanism of GPER1/GPR30 through structural and energetic analyses

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Differential expression of G-protein-coupled estrogen receptor-30 in human myometrial and uterine leiomyoma smooth muscle

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Tamoxifen has a proliferative effect in endometrial carcinoma mediated via the GPER/EGFR/ERK/cyclin D1 pathway: A retrospective study and an in vitro study

Zhang, L., Li, Y., Lan, L., Liu, R., Wu, Y., Qu, Q., & Wen, K. (2016) · Molecular and Cellular Endocrinology · doi:10.1016/j.mce.2016.08.011 · Cited by 33 · see citing works

Estrogenic transmembrane receptor of GPR30 mediates invasion and carcinogenesis by endometrial cancer cell line RL95-2

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6PPD and 6PPD Quinone Induce Endometrial Cell Dysfunction via Activating ERα and GPER at Human-Relevant Levels

Tang, L., Li, X., Zhu, S.-Y., Wan, Y.-K., Zhang, S.-K., Ma, J., Yang, Y., Chen, A., Luo, L., & Cao, L.-Y. (2025) · Environmental Science & Technology · doi:10.1021/acs.est.4c13961 · Cited by 32 · see citing works

G protein–coupled estrogen receptor 1 agonist G-1 induces cell cycle arrest in the mitotic phase, leading to apoptosis in endometriosis

Mori, T., Ito, F., Matsushima, H., Takaoka, O., Tanaka, Y., Koshiba, A., Kusuki, I., & Kitawaki, J. (2015) · Fertility and Sterility · doi:10.1016/j.fertnstert.2015.01.026 · Cited by 31 · see citing works

Signaling through non-membrane nuclear phosphoinositide binding proteins in human health and disease

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Modulation of Burst Firing of Neurons in Nucleus Reticularis of the Thalamus by GluN2C-Containing NMDA Receptors

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Neurosteroids, trigger of the LH surge

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Stimulation of GPR30 Increases Release of EMMPRIN-Containing Microvesicles in Human Uterine Epithelial Cells

Burnett, L. A., Light, M. M., Mehrotra, P., & Nowak, R. A. (2012) · The Journal of Clinical Endocrinology & Metabolism · doi:10.1210/jc.2012-2098 · Cited by 27 · see citing works

GPER modulators: Opportunity Nox on the heels of a class Akt

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Extent of Vascular Remodeling Is Dependent on the Balance Between Estrogen Receptor α and G-Protein–Coupled Estrogen Receptor

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Various types of adenomyosis and endometriosis: in search of optimal management

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Phosphatidylinositolphosphate phosphatase activities and cancer

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G-1 exhibit antidepressant effect, increase of hippocampal ERs expression and improve hippocampal redox status in aged female rats

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G protein-coupled estrogen receptor 1 as a novel regulator of blood pressure

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Immunohistochemical expression of GPR 30 in breast carcinoma of Egyptian patients: an association with immunohistochemical subtypes

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ERα17p, an ERα P295-T311 fragment, modifies the migration of breast cancer cells, through actin cytoskeleton rearrangements

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Human G protein-coupled receptor 30 is N-glycosylated and N-terminal domain asparagine 44 is required for receptor structure and activity

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The acyl chains of phosphoinositide PIP3 alter the structure and function of nuclear receptor steroidogenic factor-1

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The G protein-coupled receptor GPR30 mediates the proliferative effects induced by 17beta-estradiol and hydroxytamoxifen in endometrial cancer cells.

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The G protein-coupled receptor GPR30 mediates the proliferative effects induced by 17beta-estradiol and hydroxytamoxifen in endometrial cancer cells

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The G protein-coupled receptor GPR30 mediates the proliferative and invasive effects induced by hydroxytamoxifen in endometrial cancer cells

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The G protein-coupled receptor GPR30 mediates proliferative effects induced by 17beta estradiol and hydroxyl tamoxifen in endometrial cancer cells

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G Protein-Coupled Receptor 30 Expression Is Up-Regulated by EGF and TGFα in Estrogen Receptor α-Positive Cancer Cells

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