International Union of Pharmacology XXXVII. Nomenclature for Leukotriene and Lipoxin Receptors

Leukotrienes: Mediators of Immediate Hypersensitivity Reactions and Inflammation

Samuelsson, B. (1983) · Science · doi:10.1126/science.6301011 · Cited by 2,843

Leukotrienes and Lipoxins: Structures, Biosynthesis, and Biological Effects

Samuelsson, B., Dahlén, S.-E., Lindgren, J. Å., Rouzer, C. A., & Serhan, C. N. (1987) · Science · doi:10.1126/science.2820055 · Cited by 2,233

Leukotriene B, a potent chemokinetic and aggregating substance released from polymorphonuclear leukocytes

Ford-Hutchinson, A. W., Bray, M. A., Doig, M. V., Shipley, M. E., & Smith, M. J. H. (1980) · Nature · doi:10.1038/286264a0 · Cited by 2,060

Diversity of G Proteins in Signal Transduction

Simon, M. I., Strathmann, M. P., & Gautam, N. (1991) · Science · doi:10.1126/science.1902986 · Cited by 2,014

The PPARα–leukotriene B4 pathway to inflammation control

Devchand, P. R., Keller, H., Peters, J. M., Vazquez, M., Gonzalez, F. J., & Wahli, W. (1996) · Nature · doi:10.1038/384039a0 · Cited by 1,345

Prostaglandin D2 Selectively Induces Chemotaxis in T Helper Type 2 Cells, Eosinophils, and Basophils via Seven-Transmembrane Receptor Crth2

Hirai, H., Tanaka, K., Yoshie, O., Ogawa, K., Kenmotsu, K., Takamori, Y., Ichimasa, M., Sugamura, K., Nakamura, M., Takano, S., et al. (2001) · The Journal of Experimental Medicine · doi:10.1084/jem.193.2.255 · Cited by 1,099

Leukotrienes promote plasma leakage and leukocyte adhesion in postcapillary venules: in vivo effects with relevance to the acute inflammatory response.

Dahlén, S. E., Björk, J., Hedqvist, P., Arfors, K. E., Hammarström, S., Lindgren, J. A., & Samuelsson, B. (1981) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.78.6.3887 · Cited by 1,019

Leukotriene C: a slow-reacting substance from murine mastocytoma cells.

Murphy, R. C., Hammarström, S., & Samuelsson, B. (1979) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.76.9.4275 · Cited by 991

A G-protein-coupled receptor for leukotriene B4 that mediates chemotaxis

Yokomizo, T., Izumi, T., Chang, K., Takuwa, Y., & Shimizu, T. (1997) · Nature · doi:10.1038/42506 · Cited by 971

Characterization of the human cysteinyl leukotriene CysLT1 receptor

Lynch, K. R., O'Neill, G. P., Liu, Q., Im, D.-S., Sawyer, N., Metters, K. M., Coulombe, N., Abramovitz, M., Figueroa, D. J., Zeng, Z., et al. (1999) · Nature · doi:10.1038/21658 · Cited by 965

Leukotrienes are potent constrictors of human bronchi

Dahlén, S.-E., Hedqvist, P., Hammarström, S., & Samuelsson, B. (1980) · Nature · doi:10.1038/288484a0 · Cited by 958

Lipoxins: novel series of biologically active compounds formed from arachidonic acid in human leukocytes.

Serhan, C. N., Hamberg, M., & Samuelsson, B. (1984) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.81.17.5335 · Cited by 765

Characterization of the Human Cysteinyl Leukotriene 2 Receptor

Heise, C. E., O'Dowd, B. F., Figueroa, D. J., Sawyer, N., Nguyen, T., Im, D.-S., Stocco, R., Bellefeuille, J. N., Abramovitz, M., Cheng, R., et al. (2000) · Journal of Biological Chemistry · doi:10.1074/jbc.m003490200 · Cited by 658

Transformation of arachidonic acid by rabbit polymorphonuclear leukocytes. Formation of a novel dihydroxyeicosatetraenoic acid.

Borgeat, P., & Samuelsson, B. (1979) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(17)30120-5 · Cited by 648

Transformation of arachidonic acid and homo-gamma-linolenic acid by rabbit polymorphonuclear leukocytes. Monohydroxy acids from novel lipoxygenases

Borgeat, P., Hamberg, M., & Samuelsson, B. (1976) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(19)57008-9 · Cited by 641

The release of histamine and formation of a slow‐reacting substance (SRS‐A) during anaphylactic shock

Brocklehurst, W. E. (1960) · The Journal of Physiology · doi:10.1113/jphysiol.1960.sp006449 · Cited by 634

Comparative airway and vascular activities of leukotrienes C-1 and D in vivo and in vitro.

Drazen, J. M., Austen, K. F., Lewis, R. A., Clark, D. A., Goto, G., Marfat, A., & Corey, E. J. (1980) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.77.7.4354 · Cited by 626

Local Effects of Synthetic Leukotrienes (LTC4, LTD4, and LTB4) in Human Skin

Soter, N. A., Lewis, R. A., Corey, E. J., & Austen, K. F. (1983) · Journal of Investigative Dermatology · doi:10.1111/1523-1747.ep12531738 · Cited by 589

Metabolism of arachidonic acid in polymorphonuclear leukocytes. Structural analysis of novel hydroxylated compounds.

Borgeat, P., & Samuelsson, B. O. (1979) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(18)36026-5 · Cited by 550

A Second Leukotriene B4 Receptor, Blt2

Yokomizo, T., Kato, K., Terawaki, K., Izumi, T., & Shimizu, T. (2000) · The Journal of Experimental Medicine · doi:10.1084/jem.192.3.421 · Cited by 538

Leukotriene E4 and granulocytic infiltration into asthmatic airways

Laitinen, L. A., Haahtela, T., Vilkka, V, Lee, T. H., & Spur, B. W. (1993) · The Lancet · doi:10.1016/0140-6736(93)91073-u · Cited by 526

The human PMN leukocyte chemotactic activity of complex hydroxy-eicosatetraenoic acids (HETEs).

Goetzl, E. J., & Pickett, W. C. (1980) · The Journal of Immunology · doi:10.4049/jimmunol.125.4.1789 · Cited by 512

Arachidonic acid metabolism in polymorphonuclear leukocytes: unstable intermediate in formation of dihydroxy acids.

Borgeat, P., & Samuelsson, B. (1979) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.76.7.3213 · Cited by 470

Endogenous lipid- and peptide-derived anti-inflammatory pathways generated with glucocorticoid and aspirin treatment activate the lipoxin A4 receptor

Perretti, M., Chiang, N., La, M., Fierro, I. M., Marullo, S., Getting, S. J., Solito, E., & Serhan, C. N. (2002) · Nature Medicine · doi:10.1038/nm786 · Cited by 447

Identification of a human cDNA encoding a functional high affinity lipoxin A4 receptor.

Fiore, S., Maddox, J. F., Perez, H. D., & Serhan, C. N. (1994) · The Journal of experimental medicine · doi:10.1084/jem.180.1.253 · Cited by 436

Slow reacting substances of anaphylaxis: Identification of leukotrienes C-1 and D from human and rat sources

Lewis, R. A., Austen, K. F., Drazen, J. M., Clark, D. A., Marfat, A., & Corey, E. J. (1980) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.77.6.3710 · Cited by 431

Aspirin-triggered 15-Epi-Lipoxin A4 (LXA4) and LXA4 Stable Analogues Are Potent Inhibitors of Acute Inflammation: Evidence for Anti-inflammatory Receptors

Takano, T., Fiore, S., Maddox, J. F., Brady, H. R., Petasis, N. A., & Serhan, C. N. (1997) · The Journal of Experimental Medicine · doi:10.1084/jem.185.9.1693 · Cited by 431

Structure of slow-reacting substance of anaphylaxis from guinea-pig lung

Morris, H. R., Taylor, G. W., Piper, P. J., & Tippins, J. R. (1980) · Nature · doi:10.1038/285104a0 · Cited by 422

THE LIBERATION OF A SLOW‐REACTING SMOOTH MUSCLE‐STIMULATING SUBSTANCE IN ANAPHYLAXIS

Kellaway, C. H., & Trethewie, E. R. (1940) · Quarterly Journal of Experimental Physiology and Cognate Medical Sciences · doi:10.1113/expphysiol.1940.sp000825 · Cited by 414

Slow-reacting substances, leukotrienes C4 and D4, increase the release of mucus from human airways in vitro.

Marom, Z. M., Shelhamer, J. H., Bach, M. K., Morton, D. R., & Kaliner, M. (1982) · PubMed · doi:10.1164/arrd.1982.126.3.449 · Cited by 414

Bronchoconstrictor Effects of Leukotriene C in Humans

Weiss, J. W., Drazen, J. M., Coles, N., McFadden, E. R., Weller, P. F., Corey, E. J., Lewis, R. A., & Austen, K. F. (1982) · Science · doi:10.1126/science.7063880 · Cited by 406

Liberation of histamine and formation of lysocithin‐like substances by cobra venom

Feldberg, W., & Kellaway, C. H. (1938) · The Journal of Physiology · doi:10.1113/jphysiol.1938.sp003674 · Cited by 377

Stereospecific total synthesis of a "slow reacting substance" of anaphylaxis, leukotriene C-1

Corey, E. J., Clark, D. A., Goto, G., Marfat, A., Mioskowski, C., Samuelsson, B., & Hammarstroem, S. (1980) · Journal of the American Chemical Society · doi:10.1021/ja00524a045 · Cited by 372

The fibrinolytic receptor for urokinase activates the G protein-coupled chemotactic receptor FPRL1/LXA4R

Resnati, M., Pallavicini, I., Wang, J. M., Oppenheim, J., Serhan, C. N., Romano, M., & Blasi, F. (2002) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.022652999 · Cited by 360

Identification, Molecular Cloning, Expression, and Characterization of a Cysteinyl Leukotriene Receptor

Sarau, H. M., Ames, R. S., Chambers, J., Ellis, C., Elshourbagy, N., Foley, J. J., Schmidt, D. B., Muccitelli, R. M., Jenkins, O., Murdock, P. R., et al. (1999) · Molecular Pharmacology · doi:10.1016/s0026-895x(24)23093-5 · Cited by 345

Design of Lipoxin A4 Stable Analogs That Block Transmigration and Adhesion of Human Neutrophils

Serhan, C. N., Maddox, J. F., Petasis, N. A., Akritopoulou-Zanze, I., Papayianni, A., Brady, H. R., Colgan, S. P., & Madara, J. L. (1995) · Biochemistry · doi:10.1021/bi00044a041 · Cited by 327

Heptahelical Receptor Signaling: Beyond the G Protein Paradigm

Hall, R. A., Premont, R. T., & Lefkowitz, R. J. (1999) · The Journal of Cell Biology · doi:10.1083/jcb.145.5.927 · Cited by 325

Comparative effects of inhaled leukotriene C4, leukotriene D4, and histamine in normal human subjects.

Barnes, N. C., Piper, P. J., & Costello, J. F. (1984) · Thorax · doi:10.1136/thx.39.7.500 · Cited by 304

ATP-dependent primary active transport of cysteinyl leukotrienes across liver canalicular membrane. Role of the ATP-dependent transport system for glutathione S-conjugates.

Ishikawa, T., Müller, M., Klünemann, C., Schaub, T., & Keppler, D. (1990) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(17)30655-5 · Cited by 303

Lipoxin A4 and B4 are potent stimuli for human monocyte migration and adhesion: selective inactivation by dehydrogenation and reduction.

Maddox, J. F., & Serhan, C. N. (1996) · The Journal of experimental medicine · doi:10.1084/jem.183.1.137 · Cited by 294

Slow-reacting substances (leukotrienes) contract human airway and pulmonary vascular smooth muscle in vitro

Hanna, C. J., Bach, M. K., Pare, P. D., & Schellenberg, R. R. (1981) · Nature · doi:10.1038/290343a0 · Cited by 284

Effects of Leukotriene D on the Airways in Asthma

Griffin, M. P., Weiss, J. W., Leitch, A. G., McFadden, E. R., Corey, E. J., Austen, K. F., & Drazen, J. M. (1983) · New England Journal of Medicine · doi:10.1056/nejm198302243080807 · Cited by 284

Endothelial cell leukotriene C4 synthesis results from intercellular transfer of leukotriene A4 synthesized by polymorphonuclear leukocytes.

Feinmark, S. J., & Cannon, P. (1986) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(18)66589-5 · Cited by 280

Lipoxin biosynthesis and its impact in inflammatory and vascular events

Serhan, C. N. (1994) · Biochimica et Biophysica Acta (BBA) - Lipids and Lipid Metabolism · doi:10.1016/0005-2760(94)90185-6 · Cited by 273

Effects of LTD 4 on Human Airway Smooth Muscle Cell Proliferation, Matrix Expression, and Contraction In Vitro : Differential Sensitivity to Cysteinyl Leukotriene Receptor Antagonists

Panettieri, R. A., Tan, E. M. L., Ciocca, V., Luttmann, M. A., Leonard, T. B., & Hay, D. W. P. (1998) · American Journal of Respiratory Cell and Molecular Biology · doi:10.1165/ajrcmb.19.3.2999 · Cited by 271

Pharmacology of L-660,711 (MK-571): a novel potent and selective leukotriene D4 receptor antagonist

Jones, T. R., Zamboni, R., Belley, M., Champion, E., Charette, L., Ford-Hutchinson, A. W., Frenette, R., Gauthier, J.-Y., Leger, S., Masson, P., et al. (1989) · Canadian Journal of Physiology and Pharmacology · doi:10.1139/y89-004 · Cited by 270

Lipoxin A4 Stable Analogs Are Potent Mimetics That Stimulate Human Monocytes and THP-1 Cells via a G-protein-linked Lipoxin A4 Receptor

Maddox, J. F., Hachicha, M., Takano, T., Petasis, N. A., Fokin, V. V., & Serhan, C. N. (1997) · Journal of Biological Chemistry · doi:10.1074/jbc.272.11.6972 · Cited by 266

Lipoxin A4: A New Class of Ligand for the Ah Receptor

Schaldach, C. M., Riby, J., & Bjeldanes, L. F. (1999) · Biochemistry · doi:10.1021/bi982861e · Cited by 264

Expression of the Cysteinyl Leukotriene 1 Receptor in Normal Human Lung and Peripheral Blood Leukocytes

FIGUEROA, D. J., BREYER, R. M., DEFOE, S. K., KARGMAN, S., DAUGHERTY, B. L., WALDBURGER, K., LIU, Q., CLEMENTS, M., ZENG, Z., O'NEILL, G. P., et al. (2001) · American Journal of Respiratory and Critical Care Medicine · doi:10.1164/ajrccm.163.1.2003101 · Cited by 262

Activation of Lipoxin a4 Receptors by Aspirin-Triggered Lipoxins and Select Peptides Evokes Ligand-Specific Responses in Inflammation

Chiang, N., Fierro, I. M., Gronert, K., & Serhan, C. N. (2000) · The Journal of Experimental Medicine · doi:10.1084/jem.191.7.1197 · Cited by 260

Specific binding of leukotriene B4 to receptors on human polymorphonuclear leukocytes.

Goldman, D. W., & Goetzl, E. J. (1982) · The Journal of Immunology · doi:10.4049/jimmunol.129.4.1600 · Cited by 258

Airway Responsiveness to Leukotrienes C4 and D4 and to Methacholine in Patients with Asthma and Normal Controls

Adelroth, E., Morris, M. M., Hargreave, F. E., & O'Byrne, P. M. (1986) · New England Journal of Medicine · doi:10.1056/nejm198608213150803 · Cited by 251

Pharmacology of montelukast sodium (Singulair™), a potent and selective leukotriene D4receptor antagonist

Jones, T. R., Labelle, M., Belley, M., Champion, E., Charette, L., Evans, J., Ford-Hutchinson, A. W., Gauthier, J. Y., Lord, A., Masson, P., et al. (1995) · Canadian Journal of Physiology and Pharmacology · doi:10.1139/y95-028 · Cited by 248

Pulmonary responses to bronchoconstrictor agonists in the mouse

Martin, T. R., Gerard, N. P., Galli, S. J., & Drazen, J. M. (1988) · Journal of Applied Physiology · doi:10.1152/jappl.1988.64.6.2318 · Cited by 243

Lipoxins and novel aspirin-triggered 15-epi-lipoxins (ATL): A jungle of cell-cell interactions or a therapeutic opportunity?

Serhan, C. N. (1997) · Prostaglandins · doi:10.1016/s0090-6980(97)00001-4 · Cited by 241

Leukotriene B4: Metabolism and Signal Transduction

Yokomizo, T., Izumi, T., & Shimizu, T. (2001) · Archives of Biochemistry and Biophysics · doi:10.1006/abbi.2000.2168 · Cited by 231

Neutrophil-mediated changes in vascular permeability are inhibited by topical application of aspirin-triggered 15-epi-lipoxin A4 and novel lipoxin B4 stable analogues.

Takano, T., Clish, C. B., Gronert, K., Petasis, N., & Serhan, C. N. (1998) · Journal of Clinical Investigation · doi:10.1172/jci1578 · Cited by 230

Leukotriene B4 receptor transgenic mice reveal novel protective roles for lipoxins and aspirin-triggered lipoxins in reperfusion

Chiang, N., Gronert, K., Clish, C. B., O’Brien, J. A., Freeman, M. W., & Serhan, C. N. (1999) · Journal of Clinical Investigation · doi:10.1172/jci7016 · Cited by 218

Leukotriene D 4 : a Potent Coronary Artery Vasoconstrictor Associated with Impaired Ventricular Contraction

Michelassi, F., Landa, L., Hill, R. D., Lowenstein, E., Watkins, W. D., Petkau, A. J., & Zapol, W. M. (1982) · Science · doi:10.1126/science.6808665 · Cited by 217

Lipoxin A4 and Lipoxin B4 Inhibit Chemotactic Responses of Human Neutrophils Stimulated by Leukotriene B4 and N-Formyl-l-Methionyl-l-Leucyl-l-Phenylalanine

Lee, T. H., Horton, C. E., Kyan-Aung, U., Haskard, D., Crea, A. E. G., & Spur, B. W. (1989) · Clinical Science · doi:10.1042/cs0770195 · Cited by 215

Local and systemic delivery of a stable aspirin-triggered lipoxin prevents neutrophil recruitment in vivo

Clish, C. B., O’Brien, J. A., Gronert, K., Stahl, G. L., Petasis, N. A., & Serhan, C. N. (1999) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.96.14.8247 · Cited by 212

Identification of a Human Enterocyte Lipoxin A4 Receptor That Is Regulated by Interleukin (IL)-13 and Interferon γ and Inhibits Tumor Necrosis Factor α–induced IL-8 Release

Gronert, K., Gewirtz, A., Madara, J. L., & Serhan, C. N. (1998) · The Journal of Experimental Medicine · doi:10.1084/jem.187.8.1285 · Cited by 207

Hydroxyeicosanoids Bind to and Activate the Low Affinity Leukotriene B4 Receptor, BLT2

Yokomizo, T., Kato, K., Hagiya, H., Izumi, T., & Shimizu, T. (2001) · Journal of Biological Chemistry · doi:10.1074/jbc.m011361200 · Cited by 205

Leukotriene C4 affects pulmonary and cardiovascular dynamics in monkey

Smedegård, G., Hedqvist, P., Dahlén, S.-E., Revenäs, B., Hammarström, S., & Samuelsson, B. (1982) · Nature · doi:10.1038/295327a0 · Cited by 204

A structural homologue of the N-formyl peptide receptor. Characterization and chromosome mapping of a peptide chemoattractant receptor family.

Murphy, P. M., Ozçelik, T., Kenney, R. T., Tiffany, H. L., McDermott, D., & Francke, U. (1992) · Journal of Biological Chemistry · doi:10.1016/s0021-9258(18)42563-x · Cited by 203

The Synthetic Peptide Trp-Lys-Tyr-Met-Val-Met-NH2 Specifically Activates Neutrophils through FPRL1/Lipoxin A4 Receptors and Is an Agonist for the Orphan Monocyte-expressed Chemoattractant Receptor FPRL2

Christophe, T., Karlsson, A., Dugave, C., Rabiet, M.-J., Boulay, F., & Dahlgren, C. (2001) · Journal of Biological Chemistry · doi:10.1074/jbc.m007769200 · Cited by 202

The Molecular Characterization and Tissue Distribution of the Human Cysteinyl Leukotriene CysLT2 Receptor

Takasaki, J., Kamohara, M., Matsumoto, M., Saito, T., Sugimoto, T., Ohishi, T., Ishii, H., Ota, T., Nishikawa, T., Kawai, Y., et al. (2000) · Biochemical and Biophysical Research Communications · doi:10.1006/bbrc.2000.3140 · Cited by 201

Lipoxin (LX)A4 and Aspirin-triggered 15-epi-LXA4 Inhibit Tumor Necrosis Factor 1α–initiated Neutrophil Responses and Trafficking: Regulators of a Cytokine–Chemokine Axis

Hachicha, M., Pouliot, M., Petasis, N. A., & Serhan, C. N. (1999) · The Journal of Experimental Medicine · doi:10.1084/jem.189.12.1923 · Cited by 199

Bltr Mediates Leukotriene B4–Induced Chemotaxis and Adhesion and Plays a Dominant Role in Eosinophil Accumulation in a Murine Model of Peritonitis

Tager, A. M., Dufour, J. H., Goodarzi, K., Bercury, S. D., von Andrian, U. H., & Luster, A. D. (2000) · The Journal of Experimental Medicine · doi:10.1084/jem.192.3.439 · Cited by 195

Aspirin-Triggered Lipoxins (15-epi-LX) Are Generated by the Human Lung Adenocarcinoma Cell Line (A549)–Neutrophil Interactions and Are Potent Inhibitors of Cell Proliferation

Clària, J., Lee, M. H., & Serhan, C. N. (1996) · Molecular Medicine · doi:10.1007/bf03401642 · Cited by 192

Molecular Cloning and Characterization of a Second Human Cysteinyl Leukotriene Receptor: Discovery of a Subtype Selective Agonist

Nothacker, H.-P., Wang, Z., Zhu, Y., Reinscheid, R. K., Lin, S. H. S., & Civelli, O. (2000) · Molecular Pharmacology · doi:10.1124/mol.58.6.1601 · Cited by 191

The Physicochemical Characteristics and Purification of Slow-Reacting Substance of Anaphylaxis

Orange, R. P., Murphy, R. C., Karnovsky, M. L., & Austen, K. F. (1973) · The Journal of Immunology · doi:10.4049/jimmunol.110.3.760 · Cited by 185

Oxidoreductases in Lipoxin A4 Metabolic Inactivation

Clish, C. B., Levy, B. D., Chiang, N., Tai, H.-H., & Serhan, C. N. (2000) · Journal of Biological Chemistry · doi:10.1074/jbc.m002863200 · Cited by 184

Cysteinyl leukotriene receptor 1 is also a pyrimidinergic receptor and is expressed by human mast cells

Mellor, E. A., Maekawa, A., Austen, K. F., & Boyce, J. A. (2001) · Proceedings of the National Academy of Sciences · doi:10.1073/pnas.141221498 · Cited by 180

A novel mechanism for the Ca(2+)-sensitizing effect of protein kinase C on vascular smooth muscle: inhibition of myosin light chain phosphatase.

Masuo, M., Reardon, S., Ikebe, M., & Kitazawa, T. (1994) · The Journal of general physiology · doi:10.1085/jgp.104.2.265 · Cited by 180

Leukotrienes C4, D4 and E4: effects on human and guinea-pig cardiac preparations in vitro.

Burke, J. A., Levi, R., Guo, Z. G., & Corey, E. J. (1982) · The Journal of Pharmacology and Experimental Therapeutics · doi:10.1016/s0022-3565(25)33042-9 · Cited by 180

Targeted Disruption of the Leukotriene B4Receptor in Mice Reveals Its Role in Inflammation and Platelet-Activating Factor–Induced Anaphylaxis

Haribabu, B., Verghese, M. W., Steeber, D. A., Sellars, D. D., Bock, C. B., & Snyderman, R. (2000) · The Journal of Experimental Medicine · doi:10.1084/jem.192.3.433 · Cited by 175

Mapping of genes for the human C5a receptor (C5AR), human FMLP receptor (FPR), and two FMLP receptor homologue orphan receptors (FPRH1, FPRH2) to chromosome 19

Bao, L., Gerard, N. P., Eddy, R. L., Shows, T. B., & Gerard, C. (1992) · Genomics · doi:10.1016/0888-7543(92)90265-t · Cited by 172

Isolation of a cDNA that encodes a novel granulocyte N-formyl peptide receptor

Ye, R. D., Cavanagh, S. L., Quehenberger, O., Prossnitz, E. R., & Cochrane, C. G. (1992) · Biochemical and Biophysical Research Communications · doi:10.1016/0006-291x(92)90629-y · Cited by 168

Effect of leukotriene D4 on nasal mucosal blood flow, nasal airway resistance and nasal secretion in humans

BISGAARD, H., OLSSON, P., & BENDE, M. (1986) · Clinical & Experimental Allergy · doi:10.1111/j.1365-2222.1986.tb01960.x · Cited by 167

Selectivity of Recombinant Human Leukotriene D4, Leukotriene B4, and Lipoxin A4 Receptors with Aspirin-Triggered 15-epi-LXA4 and Regulation of Vascular and Inflammatory Responses

Gronert, K., Martinsson-Niskanen, T., Ravasi, S., Chiang, N., & Serhan, C. N. (2001) · The American Journal of Pathology · doi:10.1016/s0002-9440(10)63937-5 · Cited by 166

The mechanism of vascular leakage induced by leukotriene E4. Endothelial contraction.

Joris, I., Majno, G., Corey, E. J., & Lewis, R. A. (1987) · PubMed · Cited by 164

The effect of inhaled leukotriene D4 in humans.

Smith, L. J., Greenberger, P. A., Patterson, R., Krell, R. D., & Bernstein, P. R. (1985) · PubMed · doi:10.1164/arrd.1985.131.3.368 · Cited by 162

Pathogen-induced chemokine secretion from model intestinal epithelium is inhibited by lipoxin A4 analogs.

Gewirtz, A. T., McCormick, B., Neish, A. S., Petasis, N. A., Gronert, K., Serhan, C. N., & Madara, J. L. (1998) · Journal of Clinical Investigation · doi:10.1172/jci1339 · Cited by 158

The Effects of Lipoxin A 4 on Airway Responses in Asthmatic Subjects

Christie, P. E., Spur, B. W., & Lee, T. H. (1992) · American Review of Respiratory Disease · doi:10.1164/ajrccm/145.6.1281 · Cited by 158

IL-13 and IL-4 Up-Regulate Cysteinyl Leukotriene 1 Receptor Expression in Human Monocytes and Macrophages

Thivierge, M., Staňková, J., & Rola‐Pleszczynski, M. (2001) · The Journal of Immunology · doi:10.4049/jimmunol.167.5.2855 · Cited by 157

Comparison of leukotriene B4 and D4 effects on human eosinophil and neutrophil motility in vitro

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The Preclinical Pharmacology of ICI 204,219: A Peptide Leukotriene Antagonist

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