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Caveolae: From Cell Biology to Animal Physiology

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Cloning, expression, and characterization of a membrane progestin receptor and evidence it is an intermediary in meiotic maturation of fish oocytes

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Src Tyrosine Kinases, Gα Subunits, and H-Ras Share a Common Membrane-anchored Scaffolding Protein, Caveolin

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Identification, classification, and partial characterization of genes in humans and other vertebrates homologous to a fish membrane progestin receptor

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A corticosteroid receptor in neuronal membranes

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Orphan Nuclear Receptors: Shifting Endocrinology into Reverse

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Perception of Brassinosteroids by the Extracellular Domain of the Receptor Kinase BRI1

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Nuclear receptor ligand-binding domains: three-dimensional structures, molecular interactions and pharmacological implications

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Proximal Events in Signaling by Plasma Membrane Estrogen Receptors

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Impaired insulin secretory capacity in mice lacking a functional vitamin D receptor

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Reversal of Bone Loss in Mice by Nongenotropic Signaling of Sex Steroids

Kousteni, S., Chen, J.-R., Bellido, T., Han, L., Ali, A. A., O'Brien, C. A., Plotkin, L., Fu, Q., Mancino, A. T., Wen, Y., et al. (2002) · Science · doi:10.1126/science.1074935 · Cited by 420 · see citing works

Linkage of Rapid Estrogen Action to MAPK Activation by ERα-Shc Association and Shc Pathway Activation

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Rapid Actions of Steroid Receptors in Cellular Signaling Pathways

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CORRELATIONS BETWEEN THE CHEMICAL STRUCTURE AND THE PHARMACOLOGICAL ACTIONS OF THE STEROIDS1

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Nuclear receptor coregulators: multiple modes of modification.

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Cellular functions of plasma membrane estrogen receptors

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Nuclear-Receptor Ligands and Ligand-Binding Domains

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Identification of a Structural Determinant Necessary for the Localization and Function of Estrogen Receptor α at the Plasma Membrane

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Identification of a specific binding protein for 1 alpha,25-dihydroxyvitamin D3 in basal-lateral membranes of chick intestinal epithelium and relationship to transcaltachia.

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Functional testosterone receptors in plasma membranes of T cells

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Plasma Membrane Estrogen Receptors Are Coupled to Endothelial Nitric-oxide Synthase through Gαi

Wyckoff, M. H., Chambliss, K. L., Mineo, C., Yuhanna, I. S., Mendelsohn, M. E., Mumby, S. M., & Shaul, P. W. (2001) · Journal of Biological Chemistry · doi:10.1074/jbc.m100312200 · Cited by 282 · see citing works

Androgens increase intracellular calcium concentration and inositol 1,4,5-trisphosphate and diacylglycerol formation via a pertussis toxin-sensitive G-protein.

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Endometrial cell calcium and oestrogen action

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Testosterone stimulates intracellular calcium release and mitogen-activated protein kinases via a G protein-coupled receptor in skeletal muscle cells

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ERβ Has Nongenomic Action in Caveolae

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Antagonists Selective for Estrogen Receptor

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Vitamin D3 Metabolites Modulate Dihydropyridine-sensitive Calcium Currents in Clonal Rat Osteosarcoma Cells

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CHROMOSOMAL RECEPTOR FOR A VITAMIN D METABOLITE

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Plasma Membrane Estrogen Receptors Signal to Antiapoptosis in Breast Cancer

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Nongenomic Actions of Thyroid Hormone on the Heart

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Two Domains of the Progesterone Receptor Interact with the Estrogen Receptor and Are Required for Progesterone Activation of the c-Src/Erk Pathway in Mammalian Cells

Ballaré, C., Uhrig, M., Bechtold, T., Sancho, E., Domenico, M. D., Migliaccio, A., Auricchio, F., & Beato, M. (2003) · Molecular and Cellular Biology · doi:10.1128/mcb.23.6.1994-2008.2003 · Cited by 222 · see citing works

Target selection in drug discovery

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Membrane‐Initiated Steroid Actions and theProteins that Mediate Them

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Designing Non-Peptide Peptidomimetics in the 21st Century: Inhibitors Targeting Conformational Ensembles

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Sex hormone-binding globulin mediates steroid hormone signal transduction at the plasma membrane

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Estrogen Receptor-α Detected on the Plasma Membrane of Aldehyde-Fixed GH3/B6/F10 Rat Pituitary Tumor Cells by Enzyme-Linked Immunocytochemistry*

Norfleet, A. M., Thomas, M. L., Gametchu, B., & Watson, C. S. (1999) · Endocrinology · doi:10.1210/endo.140.8.6936 · Cited by 170 · see citing works

Crystal structure of human sex hormone‐binding globulin: steroid transport by a laminin G‐like domain

Grishkovskaya, I., Avvakumov, G. V., Sklenar, G., Dales, D. W., Hammond, G. L., & Muller, Y. A. (2000) · The EMBO Journal · doi:10.1093/emboj/19.4.504 · Cited by 170 · see citing works

1α,25-Dihydroxyvitamin D 3 Induces Vascular Smooth Muscle Cell Migration via Activation of Phosphatidylinositol 3-Kinase

Rebsamen, M. C., Sun, J., Norman, A. W., et al. (2002) · Circulation Research · doi:10.1161/01.res.0000025269.60668.0f · Cited by 164 · see citing works

The human prostate cancer cell line LNCaP bears functional membrane testosterone receptors, which increase PSA secretion and modify actin cytoskeleton

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A structural basis for the unique binding features of the human vitamin D-binding protein

Verboven, C., Rabijns, A., Maeyer, M. D., BAELEN, H. V., Bouillon, R., & Ranter, C. D. (2002) · Nature Structural Biology · doi:10.1038/nsb754 · Cited by 154 · see citing works

Molecular Mechanisms of Gating and Drug Block of Sodium Channels

Carterall, W. A. (2001) · Novartis Foundation symposium · doi:10.1002/0470846682.ch14 · Cited by 145 · see citing works

Androgen-stimulated DNA synthesis and cytoskeletal changes in fibroblasts by a nontranscriptional receptor action

Castoria, G., Lombardi, M., Barone, M. V., Bilancio, A., Domenico, M. D., Bottero, D., Vitale, F., Migliaccio, A., & Auricchio, F. (2003) · The Journal of Cell Biology · doi:10.1083/jcb.200211099 · Cited by 136 · see citing works

Testosterone induces Ca2+ influx via non‐genomic surface receptors in activated T cells

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Estradiol Signaling via Sequestrable Surface Receptors

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Antibodies to the estrogen receptor‐α modulate rapid prolactin release from rat pituitary tumor cells through plasma membrane estrogen receptors

Norfleet, A. M., Clarke, C. H., Gametchu, B., & Watson, C. S. (2000) · The FASEB Journal · doi:10.1096/fasebj.14.1.157 · Cited by 129 · see citing works

Direct Activation of Protein Kinase C by 1α,25-Dihydroxyvitamin D3

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Nuclear receptors in cell life and death

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The Classical Progesterone Receptor Associates with p42 MAPK and Is Involved in Phosphatidylinositol 3-Kinase Signaling inXenopus Oocytes

Bagowski, C. P., Myers, J. W., & Ferrell, J. E. (2001) · Journal of Biological Chemistry · doi:10.1074/jbc.m104582200 · Cited by 125 · see citing works

Stimulation of Phosphorylation of Mitogen-Activated Protein Kinase by 1α,25-Dihydroxyvitamin D3 in Promyelocytic NB4 Leukemia Cells: A Structure-Function Study*

Song, X., Bishop, J. E., Okamura, W. H., & Norman, A. W. (1998) · Endocrinology · doi:10.1210/endo.139.2.5747 · Cited by 125 · see citing works

Comparison of 6-s-cis- and 6-s-trans-Locked Analogs of 1α,25-Dihydroxyvitamin D3 Indicates That the 6-s-cis Conformation Is Preferred for Rapid Nongenomic Biological Responses and That Neither 6-s-cis- nor 6-s-trans-Locked Analogs Are Preferred for Genomic Biological Responses

Norman, A. W., Okamura, W. H., Hammond, M. W., Bishop, J. E., Dormanen, M. C., Bouillon, R., BAELEN, H. V., Ridall, A. L., Daane, E., Khoury, R., et al. (1997) · Molecular Endocrinology · doi:10.1210/mend.11.10.9993 · Cited by 123 · see citing works

Selective Modulation of Genomic and Nongenomic Androgen Responses by Androgen Receptor Ligands

Lutz, L. B., Jamnongjit, M., Yang, W., Jahani, D., Gill, A., & Hammes, S. R. (2003) · Molecular Endocrinology · doi:10.1210/me.2003-0032 · Cited by 112 · see citing works

An Insulinotropic Effect of Vitamin D Analog with Increasing Intracellular Ca2+ Concentration in Pancreatic β-Cells through Nongenomic Signal Transduction1

Kajikawa, M., Ishida, H., Fujimoto, S., Mukai, E., Nishimura, M., Fujita, J., Tsuura, Y., Okamoto, Y., Norman, A. W., & Seino, Y. (1999) · Endocrinology · doi:10.1210/endo.140.10.7025 · Cited by 110 · see citing works

Ligand–protein interactions in nuclear receptors of hormones

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Estradiol Signaling via Sequestrable Surface Receptors

Benten, W. P. M., Stephan, C., Lieberherr, M., & Wunderlich, F. T. (2001) · Endocrinology · doi:10.1210/endo.142.4.8094 · Cited by 106 · see citing works

Intracellular calcium increase and acrosome reaction in response to progesterone in human spermatozoa are correlated with in-vitro fertilization

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Progesterone Triggers a Wave of Increased Free Calcium during the Human Sperm Acrosome Reaction

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Membrane-Initiated Steroid Actions and the Proteins that Mediate Them

Watson, C. S., & Gametchu, B. (1999) · Experimental Biology and Medicine · doi:10.3181/00379727-220-44338 · Cited by 104 · see citing works

Stimulation by 1α,25(OH)2-Vitamin D3 of Whole Cell Chloride Currents in Osteoblastic ROS 17/2.8 Cells

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Effects of thyroid hormone on action potential and repolarizing currents in rat ventricular myocytes

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Coupling Gβγ-Dependent Activation to Channel Opening via Pore Elements in Inwardly Rectifying Potassium Channels

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Minireview: Genomics Versus Orphan Nuclear Receptors--A Half-Time Report

Willson, T. M., & Moore, J. T. (2002) · Molecular Endocrinology · doi:10.1210/mend.16.6.0849 · Cited by 82 · see citing works

Partial purification and biochemical characterization of a membrane glucocorticoid receptor from an amphibian brain

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Molecular tools for study of genomic and rapid signal transduction responses initiated by 1α,25(OH)2-vitamin D3

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OmpA: A Pore or Not a Pore? Simulation and Modeling Studies

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Involvement of hydrogen peroxide in the differentiation of clonal HD‐11EM cells into osteoclast‐like cells

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Retardation of Sodium Exchange in Dog Erythrocytes by Physiological Concentrations of Aldosterone, in Vitro*

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Monocytic Differentiation of Acute Promyelocytic Leukemia Cells in Response to 1,25-Dihydroxyvitamin D3 Is Independent of Nuclear Receptor Binding

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Different shapes of the steroid hormone 1α,25(OH)2-vitamin D3 act as agonists for two different receptors in the vitamin D endocrine system to mediate genomic and rapid responses☆11☆ Guest Editor: Dr. Satya Reddy, Proceedings of the First International Conference on Chemistry and Biology of Vitamin D Analogs, Brown University, Providence, RI.

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Nongenomic Mechanisms of Glucocorticoid Inhibition of Nicotine-Induced Calcium Influx in PC12 Cells: Involvement of Protein Kinase C**This work was supported by a research grant from the Natural Science Foundation of China.

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Non-classical receptors for aldosterone in plasma membranes from pig kidneys

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