Modulators of Protein–Protein Interactions

Cites (624)

Items 401–600 of 624

1. Blocking Estrogen Signaling After the Hormone: Pyrimidine-Core Inhibitors of Estrogen Receptor-Coactivator Binding
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2. Acylpyrogallols as Inhibitors of Antiapoptotic Bcl-2 Proteins
   Guozhi Tang, Zaneta Nikolovska‐Coleska, Su Qiu, Chao‐Yie Yang, Jie Guo, Shaomeng Wang · 2008 · Journal of Medicinal Chemistry
3. クリプテート発光の時間分解増幅 生物分子相互作用を追跡するための多才な技術 | 文献情報 | J-GLOBAL 科学技術総合リンクセンター
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4. (+)-Discodermolide: total synthesis, construction of novel analogues, and biological evaluation
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5. Antibody-enabled small-molecule drug discovery
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6. Context-Based Identification of Protein-Protein Interfaces and “Hot-Spot” Residues
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7. Phage selection of bicyclic peptides
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8. Stabilization of an α Helix by β‐Sheet‐Mediated Self‐Assembly of a Macrocyclic Peptide
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9. KCa3.1: target and marker for cancer, autoimmune disorder and vascular inflammation?
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10. Quantifying protein–protein interactions in high throughput using protein domain microarrays
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11. Apamin as a Template for Structure‐Based Rational Design of Potent Peptide Activators of p53
    Chong Li, Marzena Pazgier, Min Liu, Wei‐Yue Lu, Wuyuan Lu · 2009 · Angewandte Chemie International Edition
12. Alternative Inhibition of Androgen Receptor Signaling: Peptidomimetic Pyrimidines As Direct Androgen Receptor/Coactivator Disruptors
    Jillian Rebecca Gunther, A.A. Parent, John A. Katzenellenbogen · 2009 · ACS Chemical Biology
13. Small Conductance Ca2+-Activated K+ Channels as Targets of CNS Drug Development
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14. Synthesis and evaluation of anthranilic acid-based transthyretin amyloid fibril inhibitors
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15. A Synthetic Supramolecular Construct Modulating Protein Assembly in Cells
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16. A Biosensor of S100A4 Metastasis Factor Activation: Inhibitor Screening and Cellular Activation Dynamics
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17. Identification of the first non-peptidic small molecule inhibitor of the c-Abl/14-3-3 protein–protein interactions able to drive sensitive and Imatinib-resistant leukemia cells to apoptosis
    Valentina Corradi, Manuela Mancini, Fabrizio Manetti, Sara Petta, Maria Alessandra Santucci, Maurizio Botta · 2010 · Bioorganic & Medicinal Chemistry Letters
18. Toward Optimization of the Linker Substructure Common to Transthyretin Amyloidogenesis Inhibitors Using Biochemical and Structural Studies
    Steven M. Johnson, Stephen Connelly, Ian A. Wilson, Jeffery W. Kelly · 2008 · Journal of Medicinal Chemistry
19. Bcl-XL-Templated Assembly of Its Own Protein−Protein Interaction Modulator from Fragments Decorated with Thio Acids and Sulfonyl Azides
    Xiangdong Hu, Jiazhi Sun, Hong‐Gang Wang, Roman Manetsch · 2008 · Journal of the American Chemical Society
20. Catalytic Inhibitors of Topoisomerase II Differently Modulate the Toxicity of Anthracyclines in Cardiac and Cancer Cells
    Anna Jirkovská, Hana Jansová, Eliška Macková, Miloslav Macháček, Pavlína Hašková, Lucie Tichotová, Martin Štěrba, Tomáš Šimůnek · 2013 · PLoS ONE
21. SK2 Channels Are Neuroprotective for Ischemia-Induced Neuronal Cell Death
    Duane Allen, Shin Nakayama, Masayuki Kuroiwa, Takaaki Nakano, Julie Palmateer, Yasuharu Kosaka, Carmen Ballesteros, Masahiko Watanabe, Chris T. Bond, Rafael Luján et al. · 2011 · Journal of Cerebral Blood Flow & Metabolism
22. Turning a Scorpion Toxin into an Antitumor Miniprotein
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23. Synthetic mimetics of protein secondary structure domains
    Nathan T. Ross, William P. Katt, Andrew D. Hamilton · 2010 · Philosophical Transactions of the Royal Society A Mathematical Physical and Engineering Sciences
24. Design of Bcl-2 and Bcl-xL Inhibitors with Subnanomolar Binding Affinities Based upon a New Scaffold
    Haibin Zhou, Jianfang Chen, Jennifer L. Meagher, Chao‐Yie Yang, Angelo Aguilar, Liu Liu, Longchuan Bai, Xin Cong, Qian Cai, Xueliang Fang et al. · 2012 · Journal of Medicinal Chemistry
25. A Natural Product Inspired Tetrahydropyran Collection Yields Mitosis Modulators that Synergistically Target CSE1L and Tubulin
    Tobias Voigt, Claas Gerding‐Reimers, Tuyen Thi Ngoc Tran, Sabrina Bergmann, Hugo Lachance, Beate Schölermann, Andreas Brockmeyer, Petra Janning, Slava Ziegler, Herbert Waldmann · 2012 · Angewandte Chemie International Edition
26. Relative Helix−Helix Conformations in Branched Aromatic Oligoamide Foldamers
    Nicolas Delsuc, Stéphane Massip, Jean‐Michel Léger, Brice Kauffmann, Ivan Huc · 2011 · Journal of the American Chemical Society
27. Isolation of a New Plant Growth Substance with Cytokinin-like Activity
    Takeshi Sassa, T. TOJYO, Katsura Munakata · 1970 · Nature
28. Identification of the functional binding pocket for compounds targeting small-conductance Ca2+-activated potassium channels
    Miao Zhang, John M. Pascal, Marcel René Schumann, Roger S. Armen, Ji-Fang Zhang · 2012 · Nature Communications
29. Kinetic target-guided synthesis
    Xiangdong Hu, Roman Manetsch · 2010 · Chemical Society Reviews
30. Ordering of the N-Terminus of Human MDM2 by Small Molecule Inhibitors
    Klaus Michelsen, John B. Jordan, Jeffrey K. Lewis, Alexander M. Long, Evelyn Yang, Yosup Rew, Jing Zhou, Peter S. Yakowec, Paul D. Schnier, Xin Yun Huang et al. · 2012 · Journal of the American Chemical Society
31. Modulating Protein–Protein Interactions with Small Molecules: The Importance of Binding Hotspots
    Thangudu, Ratna Rajesh, Bryant, Stephen H., Panchenko, Anna R., Madej, Thomas · 2012 · Journal of Molecular Biology
32. Cotylenin A, a Plant-Growth Regulator, Induces the Differentiation in Murine and Human Myeloid Leukemia Cells
    Ken‐ichi Asahi, Yoshio Honma, Kaoru Hazeki, Takeshi Sassa, Yuzuru Kubohara, Akira Sakurai, Nobutaka Takahashi · 1997 · Biochemical and Biophysical Research Communications
33. Modular α-Helical Mimetics with Antiviral Activity against Respiratory Syncitial Virus
    Nicholas E. Shepherd, Huy N. Hoang, Vishal S. Desai, Éric Letouzé, Paul R. Young, David P. Fairlie · 2006 · Journal of the American Chemical Society
34. β-Peptides with improved affinity for hDM2 and hDMX
    Elizabeth A. Harker, Douglas S. Daniels, Danielle A. Guarracino, Alanna Schepartz · 2009 · Bioorganic & Medicinal Chemistry
35. The p53-MDM2/MDMX axis – A chemotype perspective
    Kareem Khoury, Grzegorz M. Popowicz, Tad A. Holak, Alexander S. S. Dömling · 2011 · MedChemComm
36. High-Throughput Screening AlphaScreen Assay for Identification of Small-Molecule Inhibitors of Ubiquitin E3 Ligase SCFSkp2-Cks1
    Ungermannova, Dana, Lee, Junglim, Zhang, Gan, Dallmann, H. Garry, McHenry, Charles S., Liu, Xuedong · 2013 · SLAS Discovery
37. A Substructure Combination Strategy To Create Potent and Selective Transthyretin Kinetic Stabilizers That Prevent Amyloidogenesis and Cytotoxicity
    Sungwook Choi, Natàlia Reixach, Stephen Connelly, Steven M. Johnson, Ian A. Wilson, Jeffery W. Kelly · 2009 · Journal of the American Chemical Society
38. Targeting SKCa Channels in Cancer: Potential New Therapeutic Approaches
    Alban Girault, Jean‐Pierre Haelters, Marie Potier‐Cartereau, Aurélie Chantôme, Paul‐Alain Jaffrès, Philippe Bougnoux, Virginie Joulin, Christophe Vandier · 2012 · Current Medicinal Chemistry
39. Thioether side chain cyclization for helical peptide formation: inhibitors of estrogen receptor–coactivator interactions
    Galande, A.K., Bramlett, K.S., Burris, T.P., Wittliff, J.L., Spatola, A.F. · 2004 · The Journal of Peptide Research
40. Development of Peptide Antagonists for the Androgen Receptor Using Combinatorial Peptide Phage Display
    Ching‐yi Chang, Jennifer Abdo, Tanya Hartney, Donald Patrick McDonnell · 2005 · Molecular Endocrinology
41. Enhancement of α-Helix Mimicry by an α/β-Peptide Foldamer via Incorporation of a Dense Ionic Side-Chain Array
    Lisa M. Johnson, D.E. Mortenson, Hyun Gi Yun, W. Seth Horne, Thomas J. Ketas, Min Lu, John P. Moore, Samuel H. Gellman · 2012 · Journal of the American Chemical Society
42. Exploring Drug Target Flexibility Using in Situ Click Chemistry: Application to a Mycobacterial Transcriptional Regulator
    Nicolas Willand, Matthieu Desroses, Patrick Toto, Bertrand Dirié, Zoé Lens, Vincent Villeret, Prakash Rucktooa, Camille Locht, Alain R. Baulard, Benoit P. Deprez · 2010 · ACS Chemical Biology
43. The translation inhibitor pateamine A prevents cachexia-induced muscle wasting in mice
    Sergio Di Marco, Anne Cammas, Xian Jin Lian, Erzsébet Nagy Kovács, Jennifer F. Ma, Derek T. Hall, Rachid Mazrouï, John Richardson, Jerry Pelletier, Imed‐Eddine Gallouzi · 2012 · Nature Communications
44. Eukaryotic ribosome display with in situ DNA recovery
    Mingyue He, Michael Taussig · 2007 · Nature Methods
45. In Silico Improvement of β3-Peptide Inhibitors of p53•hDM2 and p53•hDMX
    Julien Michel, Elizabeth A. Harker, Julian Tirado‐Rives, William L. Jorgensen, Alanna Schepartz · 2009 · Journal of the American Chemical Society
46. Trapping of palindromic ligands within native transthyretin prevents amyloid formation
    Simon Erik Kolstoe, Palma Patrizia Mangione, Vittorio Bellotti, Graham W. Taylor, Glenys A. Tennent, Stéphanie Deroo, Angus J. Morrison, Alexander J. A. Cobb, Anthony G. Coyne, Margaret G. McCammon et al. · 2010 · Proceedings of the National Academy of Sciences
47. Cucurbit[8]uril-mediated protein homotetramerization
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48. Technologies for the Synthesis of mRNA-Encoding Libraries and Discovery of Bioactive Natural Product-Inspired Non-Traditional Macrocyclic Peptides
    Kenichiro Ito, Toby Passioura, Hiroaki Suga · 2013 · Molecules
49. Structure‐Guided Rational Design of α/β‐Peptide Foldamers with High Affinity for BCL‐2 Family Prosurvival Proteins
    Brian James Smith, Erinna F. Lee, James W. Checco, Marco Evangelista, Samuel H. Gellman, Walter Douglas Fairlie · 2013 · ChemBioChem
50. Diverted total synthesis: Preparation of a focused library of latrunculin analogues and evaluation of their actin-binding properties
    Alois Fürstner, Douglas T. Kirk, Michaël D. B. Fenster, Christophe Aïssa, Dominic De Souza, Oliver Müller · 2005 · Proceedings of the National Academy of Sciences
51. Diverted Total Synthesis Leads to the Generation of Promising Cell-Migration Inhibitors for Treatment of Tumor Metastasis: In vivo and Mechanistic Studies on the Migrastatin Core Ether Analog
    Thórdur Óskarsson, Pavel Nagorny, Isaac J. Krauss, Lucy Pérez, Mihirbaran Mandal, Guangli Yang, Ouathek Ouerfelli, Danhua Xiao, Malcolm A.S. Moore, Joan Massagué et al. · 2010 · Journal of the American Chemical Society
52. Modulation of Cellular Apoptosis with Apoptotic Protease-Activating Factor 1 (Apaf-1) Inhibitors
    Laura Mondragón, Mar Orzáez, Glòria Sanclimens, Alejandra Moure, Ana Armiñán, Pilar Sepúlveda, Ángel Messeguer, Maria Jesus Vicent, Enríque Pérez‐Payá · 2008 · Journal of Medicinal Chemistry
53. NMR Strategy for Unraveling Structures of Bioactive Sponge-Derived Oxy-polyhalogenated Diphenyl Ethers
    Laurent Calcul, Raymond Kwok Kei Chow, Allen G. Oliver, Karen Tenney, Kimberly N. White, Alexander W. Wood, Catherine Fiorilla, Phillip Crews · 2009 · Journal of Natural Products
54. Selective Chemical Imaging of Static Actin in Live Cells
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55. Discovery of protein–protein binding disruptors using multi-component condensations small molecules
    Karim Bedjeguelal, Hugues Bienaymé, Antoine Dumoulin, Stéphane Poigny, Philippe Schmitt, Eric Tam · 2006 · Bioorganic & Medicinal Chemistry Letters
56. EF hands at the N-lobe of calmodulin are required for both SK channel gating and stable SK–calmodulin interaction
    Weiyan Li, David Brent Halling, Amelia Weber Hall, Richard W. Aldrich · 2009 · The Journal of General Physiology
57. Effects of combined treatment with rapamycin and cotylenin A, a novel differentiation-inducing agent, on human breast carcinoma MCF-7 cells and xenografts
    Takashi Kasukabe, Junko Okabe‐Kado, Nobuo Kato, Takeshi Sassa, Yoshio Honma · 2005 · Breast Cancer Research
58. Structural Basis of Bcl‐x L Recognition by a BH3‐Mimetic α/β‐Peptide Generated by Sequence‐Based Design
    Erinna F. Lee, Brian James Smith, W. Seth Horne, Kelsey N. Mayer, Marco Evangelista, Peter M. Colman, Samuel H. Gellman, Walter Douglas Fairlie · 2011 · ChemBioChem
59. Rational Design of Small-Molecule Inhibitors for β-Catenin/T-Cell Factor Protein–Protein Interactions by Bioisostere Replacement
    Binxun Yu, Zheng Huang, Min Zhang, Darren R. Dillard, Haitao Ji · 2012 · ACS Chemical Biology
60. Probing the Role of Backbone Hydrogen Bonds in Protein–Peptide Interactions by Amide-to-Ester Mutations
    Eildal, Jonas N. N., Hultqvist, Greta, Balle, Thomas, Stuhr-Hansen, Nicolai, Padrah, Shahrokh, Gianni, Stefano, Strømgaard, Kristian, Jemth, Per · 2013 · Journal of the American Chemical Society
61. In vivo characterisation of the small-conductance KCa (SK) channel activator 1-ethyl-2-benzimidazolinone (1-EBIO) as a potential anticonvulsant
    Neil J. Anderson, Scott Slough, William P. Watson · 2006 · European Journal of Pharmacology
62. Synthesis of a Phosphoserine Mimetic Prodrug with Potent 14-3-3 Protein Inhibitory Activity
    Allison A. Arrendale, Keunho J. Kim, Jun Young Choi, Wěi Li, Robert L. Geahlen, Richard F. Borch · 2012 · Chemistry & Biology
63. Paclitaxel from Primary Taxanes: A Perspective on Creative Invention in Organozirconium Chemistry
    Bruce Ganem, Roland R. Franke · 2007 · The Journal of Organic Chemistry
64. Ribosome-display technology: applications for directed evolution of functional proteins
    Xianghua Yan, XU Zi-rong · 2006 · Drug Discovery Today
65. In Vitro Selection of Multiple Libraries Created by Genetic Code Reprogramming To Discover Macrocyclic Peptides That Antagonize VEGFR2 Activity in Living Cells
    Takashi Kawakami, Takahiro Ishizawa, Tomoshige Fujino, Patrick Reid, Hiroaki Suga, Hiroshi Murakami · 2013 · ACS Chemical Biology
66. Synthesis and biological evaluation of guanylhydrazone coactivator binding inhibitors for the estrogen receptor
    Andrew L. LaFrate, Jillian Rebecca Gunther, Kathryn E. Carlson, John A. Katzenellenbogen · 2008 · Bioorganic & Medicinal Chemistry
67. A Host-Induced Intramolecular Charge-Transfer Complex and Light-Driven Radical Cation Formation of a Molecular Triad with Cucurbit[8]uril
    Dapeng Zou, Samir Andersson, Rong Zhang, Shiguo Sun, Björn Åkermark, Licheng Sun · 2008 · The Journal of Organic Chemistry
68. Substrate-Dependent Targeting of Eukaryotic Translation Initiation Factor 4A by Pateamine A: Negation of Domain-Linker Regulation of Activity
    Woon‐Kai Low, Yongjun Dang, Shridhar Bhat, Daniel Romo, Jun O. Liu · 2007 · Chemistry & Biology
69. β-Hairpin protein epitope mimetic technology in drug discovery
    Daniel Obrecht, Éric Chevalier, Kerstin Moehle, John A. Robinson · 2011 · Drug Discovery Today Technologies
70. Towards the systematic exploration of chemical space
    Mark Dow, Martin Fisher, THOMAS N. JAMES, Francesco Marchetti, Adam S. Nelson · 2011 · Organic & Biomolecular Chemistry
71. Cucurbit[8]uril induced heterodimerization of methylviologen and naphthalene functionalized proteins
    Dana A. Uhlenheuer, Jacqui F. Young, Hoang Duc Nguyen, Marcel Scheepstra, Luc Brunsveld · 2011 · Chemical Communications
72. Hydrophobic Binding Hot Spots of Bcl-xL Protein−Protein Interfaces by Cosolvent Molecular Dynamics Simulation
    Yang, Chao-Yie, Wang, Shaomeng · 2011 · ACS Medicinal Chemistry Letters
73. Transformation of Low-Affinity Lead Compounds into High-Affinity Protein Capture Agents
    M. Muralidhar Reddy, Kiran Bachhawat‐Sikder, Thomas J. Kodadek · 2004 · Chemistry & Biology
74. Phosphopeptide‐Dependent Labeling of 14–3–3 ζ Proteins by Fusicoccin‐Based Fluorescent Probes
    Michiko Takahashi, Akie Kawamura, Nobuo Kato, Tsuyoshi Nishi, Itaru Hamachi, Junko Ohkanda · 2011 · Angewandte Chemie International Edition
75. Calix[4]arene-based conical-shaped ligands for voltage-dependent potassium channels
    Vera Martos, Sarah C. Bell, Eva Santos, Ehud Y. Isacoff, Dirk H. Trauner, Javier de Mendoza · 2009 · Proceedings of the National Academy of Sciences
76. Principles, implementation, and application of biology-oriented synthesis (BIOS)
    Wolfram Wilk, Tobias J. Zimmermann, Markus Kaiser, Herbert Waldmann · 2009 · Biological Chemistry
77. Sekikaic Acid and Lobaric Acid Target a Dynamic Interface of the Coactivator CBP/p300
    Chinmay Y. Majmudar, Jonas Westergaard Højfeldt, Carl-Johan Arewång, William C. K. Pomerantz, Jessica K. Gagnon, Pamela J. Schultz, Laura C. Cesa, Conor H. Doss, Steven P. Rowe, Víctor Vásquez et al. · 2012 · Angewandte Chemie International Edition
78. Stereochemical and Skeletal Diversity Arising from Amino Propargylic Alcohols
    Daniela Pizzirani, Taner Kaya, Paul A. Clemons, Stuart L. Schreiber · 2010 · Organic Letters
79. Synthesis of Unprecedented Scaffold Diversity
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80. Skeletally Diverse Small Molecules Using a Build/Couple/Pair Strategy
    Takuya Uchida, Manuela Rodriquez, Stuart L. Schreiber · 2009 · Organic Letters
81. Advantages of mRNA display selections over other selection techniques for investigation of protein–protein interactions
    Hui Wang, Rihe Liu · 2011 · Expert Review of Proteomics
82. Very Strong Binding of Lithocholic Acid to β-Cyclodextrin
    Zhiwei Yang, Ronald Breslow · 1997 · Tetrahedron Letters
83. Current Screens Based on the AlphaScreen™ Technology for Deciphering Cell Signalling Pathways
    Saı̈d Taouji, Sophie Dahan, Roger Bossé, Éric Chevet · 2009 · Current Genomics
84. Metastasis-Inducing S100A4 Protein: Implication in Non-Malignant Human Pathologies
    Mariam Grigorian, Noona S. Ambartsumian, Eugene M. Lukanidin · 2008 · Current Molecular Medicine
85. Nuclear Receptors as Drug Targets
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86. Setting Up a Bioluminescence Resonance Energy Transfer High throughput Screening Assay to Search for Protein/Protein Interaction Inhibitors in Mammalian Cells
    Couturier, Cyril, Deprez, Benoit · 2012 · Frontiers in Endocrinology
87. Cell‐Permeable β‐Peptide Inhibitors of p53/hDM2 Complexation
    Elizabeth A. Harker, Alanna Schepartz · 2009 · ChemBioChem
88. Prieurianin/endosidin 1 is an actin‐stabilizing small molecule identified from a chemical genetic screen for circadian clock effectors in Arabidopsis thaliana
    Réka Tóth, Claas Gerding‐Reimers, Michael J. Deeks, Sascha Menninger, Rafael Martínez-Gallegos, Isabella A. Nougalli Tonaco, Katja Hübel, Patrick J. Hussey, Herbert Waldmann, George Coupland · 2012 · The Plant Journal
89. Inhibitors of Difficult Protein–Protein Interactions Identified by High-Throughput Screening of Multiprotein Complexes
    Laura C. Cesa, Srikanth Patury, Tomoko Komiyama, Atta Ahmad, Erik R. P. Zuiderweg, Jason E. Gestwicki · 2013 · ACS Chemical Biology
90. Screening of Protein–Protein Interaction Modulators via Sulfo-Click Kinetic Target-Guided Synthesis
    Sameer S. Kulkarni, Xiangdong Hu, Kenichiro Doi, Hong‐Gang Wang, Roman Manetsch · 2011 · ACS Chemical Biology
91. High-throughput screening for modulators of protein–protein interactions: use of photonic crystal biosensors and complementary technologies
    James T. Heeres, Paul J. Hergenrother · 2010 · Chemical Society Reviews
92. 2-O-Alkylated para-benzamide α-helix mimetics: the role of scaffold curvature
    Valeria Azzarito, Panchami Prabhakaran, Alice I. Bartlett, Natasha S. Murphy, Michaele J. Hardie, Colin A. Kilner, Thomas A. Edwards, Stuart L. Warriner, Andrew John Wilson · 2012 · Organic & Biomolecular Chemistry
93. Differentiation of human acute myeloid leukaemia cells in primary culture in response to cotylenin A, a plant growth regulator
    Kazunari Yamada, Yoshio Honma, Ken‐ichi Asahi, Takashi Sassa, Ken‐ichiro Hino, Shigeru Tomoyasu · 2001 · British Journal of Haematology
94. Exhaustive Fluorine Scanning toward Potent p53–Mdm2 Antagonists
    Huang, Yijun, Wolf, Siglinde, Koes, David, Popowicz, Grzegorz M., Camacho, Carlos J., Holak, Tad A., Dömling, Alexander · 2012 · ChemMedChem
95. Bivalent Enzyme Inhibitors Discovered Using Dynamic Covalent Chemistry
    Alexandra Clipson, Venugopal T. Bhat, Iain W. McNae, Anne M. Caniard, Dominic J. Campopiano, Michael F. Greaney · 2012 · Chemistry - A European Journal
96. The State of the Art of Chemical Biology
    Karl‐Heinz Altmann, Johannes Büchner, Horst Kessler, François Diederich, Bernhard Kräutler, Stephen J. Lippard, Rob M. J. Liskamp, Klaus Müller, Elizabeth M. Nolan, Bruno Samorı̀ et al. · 2008 · ChemBioChem
97. Design and modular parallel synthesis of a MCR derived α-helix mimetic protein–protein interaction inhibitor scaffold
    Walfrido Antuch, Sanjay Menon, Quin‐Zene Chen, Yingchun Lu, Sukumar Sakamuri, Barbara Beck, Vesna Schauer-Vukašinović, Seema Agarwal, Sibylle Hess, Alexander S. S. Dömling · 2006 · Bioorganic & Medicinal Chemistry Letters
98. Dioxygenases, Key Enzymes to Determine the Aglycon Structures of Fusicoccin and Brassicicene, Diterpene Compounds Produced by Fungi
    Yusuke Ono, Atsushi Minami, Motoyoshi Noike, Yusuke Higuchi, Tomonobu Toyomasu, Takeshi Sassa, Nobuo Kato, Tohru Dairi · 2011 · Journal of the American Chemical Society
99. Discovery of a novel 5-carbonyl-1H-imidazole-4-carboxamide class of inhibitors of the HIV-1 integrase–LEDGF/p75 interaction
    Serrao, Erik, Xu, Zhong-Liang, Debnath, Bikash, Christ, Frauke, Debyser, Zeger, Long, Ya-Qiu, Neamati, Nouri · 2013 · Bioorganic & Medicinal Chemistry
100. A conceptual framework for analysing and planning synthetic approaches to diverse lead-like scaffolds
     Paul MacLellan, Adam S. Nelson · 2013 · Chemical Communications
101. Comprehensive Experimental and Computational Analysis of Binding Energy Hot Spots at the NF-κB Essential Modulator/IKKβ Protein–Protein Interface
     Golden, Mary S., Cote, Shaun M., Sayeg, Marianna, Zerbe, Brandon S., Villar, Elizabeth A., Beglov, Dmitri, Sazinsky, Stephen L., Georgiadis, Rosina M., Vajda, Sandor, Kozakov, Dima et al. · 2013 · Journal of the American Chemical Society
102. Identifying Modulators of Protein−Protein Interactions Using Photonic Crystal Biosensors
     James T. Heeres, Seok-Ho Kim, Benjamin J. Leslie, Erich A. Lidstone, Brian T. Cunningham, Paul J. Hergenrother · 2009 · Journal of the American Chemical Society
103. Discovery of Small-Molecule Modulators of the Sonic Hedgehog Pathway
     Giannina I. Schaefer, José R. Perez, Jeremy R. Duvall, Benjamin Z. Stanton, Alykhan F. Shamji, Stuart L. Schreiber · 2013 · Journal of the American Chemical Society
104. Development of a High-Throughput Screening Assay for Inhibitors of Aggrecan Cleavage Using Luminescent Oxygen Channeling (AlphaScreen™)
     Jane Peppard, Joseph Fraser Glickman, Yang He, Shou‐Ih Hu, John Doughty, RONALD L. GOLDBERG · 2003 · SLAS DISCOVERY
105. NMR Solution Structure of a Photoswitchable Apoptosis Activating Bak Peptide Bound to Bcl-x_L
     Wysoczanski, Piotr, Mart, Robert J., Loveridge, E. Joel, Williams, Christopher, Whittaker, Sara B.-M., Crump, Matthew P., Allemann, Rudolf K. · 2012 · Journal of the American Chemical Society
106. Virtual screening and experimental validation reveal novel small-molecule inhibitors of 14-3-3 protein–protein interactions
     Philipp Thiel, Lars Röglin, Nicole Meissner, Sven Hennig, Oliver Kohlbacher, Christian Ottmann · 2013 · Chemical Communications
107. Direct targeting of β-catenin: Inhibition of protein–protein interactions for the inactivation of Wnt signaling
     Hahne, Gernot, Grossmann, Tom N. · 2013 · Bioorganic & Medicinal Chemistry
108. Inducing α-Helices in Short Oligopeptides through Binding by an Artificial Hydrophobic Cavity
     Dolain, Christel, Hatakeyama, Yoshiyuki, Sawada, Tomohisa, Tashiro, Shohei, Fujita, Makoto · 2010 · Journal of the American Chemical Society
109. Supramolecular Control of Split-GFP Reassembly by Conjugation of β-Cyclodextrin and Coumarin Units
     Seiji Sakamoto, Kazuaki Kudo · 2008 · Journal of the American Chemical Society
110. Natural product inhibitors of protein–protein interactions mediated by Src-family SH2 domains
     Bianca Sperl, Markus H. J. Seifert, Thorsten Berg · 2009 · Bioorganic & Medicinal Chemistry Letters
111. A Scaffold‐Tree‐Merging Strategy for Prospective Bioactivity Annotation of γ‐Pyrones
     Stefan Wetzel, Wolfram Wilk, Samy Chammaa, Bianca Sperl, Anke Gundula Roth, Aybike Yektaoğlu, Steffen Renner, Thorsten Berg, Christoph Arenz, Athanassios Giannis et al. · 2010 · Angewandte Chemie International Edition
112. The Nuclear Receptor-Coactivator Interaction Surface as a Target for Peptide Antagonists of the Peroxisome Proliferator-Activated Receptors
     Niharika B. Mettu, Thomas B. Stanley, Mary A. Dwyer, Michelle S. Jansen, John E. Allen, Julie M. Hall, Donald Patrick McDonnell · 2007 · Molecular Endocrinology
113. Structure and Function of Benzoylurea‐Derived α‐Helix Mimetics Targeting the Bcl‐xL/Bak Binding Interface
     Johanna M. Rodriguez, Nathan T. Ross, William P. Katt, Deepali Dhar, Gui‐in Lee, Andrew D. Hamilton · 2009 · ChemMedChem
114. End-capped α-helices as modulators of protein function
     Mahon, Andrew B., Arora, Paramjit S. · 2012 · Drug Discovery Today: Technologies
115. Biosynthetic medicinal chemistry of natural product drugs
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