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Computational modeling and biological validation of novel non-steroidal ligands for the cholesterol recognition/interaction amino acid consensus (CRAC) motif of the mitochondrial translocator protein (TSPO)

Midzak, A. S., Akula, N., Rone, M. B., & Papadopoulos, V. (2015) · Pharmacological Research · doi:10.1016/j.phrs.2015.03.023 · Cited by 20 · see citing works

The novel dual-mechanism Kv7 potassium channel/TSPO receptor activator GRT-X is more effective than the Kv7 channel opener retigabine in the 6-Hz refractory seizure mouse model

Bloms-Funke, P., Bankstahl, M., Bankstahl, J., Kneip, C., Schröder, W., & Löscher, W. (2022) · Neuropharmacology · doi:10.1016/j.neuropharm.2021.108884 · Cited by 19 · see citing works

Pharmacological modulation of TSPO in microglia/macrophages and neurons in a chronic neurodegenerative model of prion disease

Vicente-Rodríguez, M., Mancuso, R., Peris-Yague, A., Simmons, C., NIMA Consortium, Wlazly, D., Dickinson, A., Foster, A., Knight, C., Leckey, C., et al. (2023) · Journal of Neuroinflammation · doi:10.1186/s12974-023-02769-y · Cited by 17 · see citing works

Progress report on new antiepileptic drugs: A summary of the Sixteenth Eilat Conference on New Antiepileptic Drugs and Devices (<scp>EILAT XVI</scp>): I. Drugs in preclinical and early clinical development

Bialer, M., Johannessen, S. I., Koepp, M. J., Levy, R. H., Perucca, E., Perucca, P., Tomson, T., & White, H. S. (2022) · Epilepsia · doi:10.1111/epi.17373 · Cited by 17 · see citing works

TSPO ligands prevent the proliferation of vascular smooth muscle cells and attenuate neointima formation through AMPK activation

Wu, L.-P., Gong, Z.-F., Wang, H., Zhou, Z.-S., Zhang, M.-M., Liu, C., Ren, H.-M., Yang, J., Han, Y., & Zeng, C.-Y. (2020) · Acta Pharmacologica Sinica · doi:10.1038/s41401-019-0293-x · Cited by 12 · see citing works

Translocator Protein Ligands as Promising Therapeutic Tools for Anxiety Disorders

Taliani, S., Settimo, F. D., Pozzo, E. D., Chelli, B., & Martini, C. (2009) · Current Medicinal Chemistry · doi:10.2174/092986709789057653 · Cited by 39 · see citing works

Translocator Protein as a Promising Target for Novel Anxiolytics

Costa, B., Pozzo, E. D., & Martini, C. (2012) · Current Topics in Medicinal Chemistry · doi:10.2174/156802612799078720 · Cited by 41 · see citing works

Enhancing neurosteroid synthesis – Relationship to the pharmacology of translocator protein (18 kDa) (TSPO) ligands and benzodiazepines

Wolf, L., Bauer, A., Melchner, D., Hallof-Buestrich, H., Stoertebecker, P., Haen, E., Kreutz, M., Sarubin, N., Milenkovic, V. M., Wetzel, C. H., et al. (2015) · Pharmacopsychiatry · doi:10.1055/s-0035-1558003 · Cited by 27 · see citing works

Cytoprotective effects of paeoniflorin are associated with translocator protein 18 kDa

Qiu, Z.-K., Liu, X., Tang, D., Zhang, Z., Fan, Q., Pan, Y., Chen, Y., Huang, M., Zhu, T., Wang, Y., et al. (2018) · Biomedicine & Pharmacotherapy · doi:10.1016/j.biopha.2018.07.112 · Cited by 4 · see citing works

Translocator protein (18kDa) TSPO: a new diagnostic or therapeutic target for stress-related disorders?

Rupprecht, R., Wetzel, C. H., Dorostkar, M. M., Herms, J. W., Albert, N. L., Schwarzbach, J. V., Schumacher, M., & Neumann, I. D. (2022) · Molecular Psychiatry · doi:10.1038/s41380-022-01561-3 · Cited by 61 · see citing works